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9SDI image
Focal Adhesion Kinase Catalytic Domain In Complex With 6-(1H-Pyrazol-4-Yl)-Nicotinic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.53 Å Release Date: 2025-12-31
Classification: TRANSFERASE
Ligands: SO4, A1JNJ

9F0I image
Human Cyclophilin D In Complex With Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.40 Å Release Date: 2025-04-30
Classification: ISOMERASE
Ligands: A1H8Q

8CHF image
Cryo-Em Structure Of Craf:14-3-3:Mek1
Organism: Homo sapiens, Spodoptera frugiperda
Method: ELECTRON MICROSCOPY
Resolution:4.25 Å Release Date: 2024-02-21
Classification: STRUCTURAL PROTEIN
Ligands: 29L

8CPD image
Cryo-Em Structure Of Craf Dimer With 14:3:3
Organism: Homo sapiens, Spodoptera frugiperda
Method: ELECTRON MICROSCOPY
Release Date: 2024-02-21
Classification: CYTOKINE

8AU3 image
C-Met Y1234E,Y1235E Mutant In Complex With Tepotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.26 Å Release Date: 2023-09-06
Classification: TRANSFERASE
Ligands: 3E8, PG4, PEG

8AU5 image
C-Met F1200I Mutant In Complex With Tepotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.72 Å Release Date: 2023-09-06
Classification: TRANSFERASE
Ligands: 3E8, EDO, CL

8AW1 image
C-Met Y1235D Mutant In Complex With Tepotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.14 Å Release Date: 2023-09-06
Classification: TRANSFERASE
Ligands: 3E8

7ZDN image
Human Cyclophilin D In Complex With Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.55 Å Release Date: 2023-04-19
Classification: ISOMERASE
Ligands: IU0

7ZKS image
Srpk1 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.28 Å Release Date: 2023-02-22
Classification: TRANSFERASE
Ligands: IXQ, CL

7ZKX image
Srpk2 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.06 Å Release Date: 2023-02-22
Classification: TRANSFERASE
Ligands: IXQ, SO4, EDO, NO3, ACT

7ZW8 image
Identification Of M4205 A Highly Selective Inhibitor Of Ckit Mutations For Unresectable Metastatic Or Recurrent Gist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.12 Å Release Date: 2023-02-22
Classification: TRANSFERASE
Ligands: K3R

7ZY6 image
Identification Of M4205 A Highly Selective Inhibitor Of Ckit Mutations For Unresectable Metastatic Or Recurrent Gist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.09 Å Release Date: 2023-02-22
Classification: TRANSFERASE
Ligands: KCI

7R2H image
0.79A Resolution Structure Of Dmso Bound Cyclophilin D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:0.79 Å Release Date: 2023-02-15
Classification: ISOMERASE
Ligands: DMS

7R2I image
Human Cyclophilin D In Complex With Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.31 Å Release Date: 2023-02-15
Classification: ISOMERASE
Ligands: DMS, UPZ, 1PE

7R2J image
Human Cyclophilin D In Complex With N-(4-Aminophenyl)-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.26 Å Release Date: 2023-02-15
Classification: ISOMERASE
Ligands: V0Z, DMS

7R2L image
Human Cyclophilin D In Complex With N-(4-Aminophenyl)-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.10 Å Release Date: 2023-02-15
Classification: ISOMERASE
Ligands: UX5, DMS, PG4

7PMT image
Human Cyclophilin D In Complex With N-[(5-Ethyl-4-Oxo-1,2,3,4,5,6- Hexahydro-1,5-Benzodiazocin-8-Yl)Methyl]-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:0.98 Å Release Date: 2022-09-14
Classification: ISOMERASE
Ligands: DMS, 7UO

7OGI image
Human Cyclophilin D In Complex With N-(5-Ethyl-4-Oxo-1,2,3,4,5,6-Hexahydro-1,5-Benzodiazocin-8-Yl)-7Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.01 Å Release Date: 2022-06-01
Classification: ISOMERASE
Ligands: VDH, DMS, PG4

7NI4 image
Human Atm Kinase Domain With Bound M4076 Inhibitor
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-09-01
Classification: SIGNALING PROTEIN
Ligands: ZN, UGK

7NI5 image
Human Atm Kinase With Bound Inhibitor Ku-55933
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-09-01
Classification: SIGNALING PROTEIN
Ligands: UF8, ZN
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