Search Count: 74
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Hiv-1 Nef Sf2 Core Domain Bound To The Human Hck Sh3 Domain
Organism: Hiv-1 m:b_arv2/sf2, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2026-07-22 Classification: VIRAL PROTEIN Ligands: EDO, NO3 |
Organism: Hiv-1 m:b_arv2/sf2, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: EDO, NO3
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Crystal Structure Of Human Wild-Type Fgr Sh3-Sh2-Linker Domains.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: GOL
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Crystal Structure Of Human Fgr Sh3-Sh2-High Affinity Linker Mutant 1 (Hal1) Domains.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: GOL, PEG
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Crystal Structure Of Human Fgr Sh3-Sh2-High Affinity Linker Mutant 2 (Hal2) Domains.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: SO4, GOL, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: SO4, GOL, FLC
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Crystal Structure Of Human Fgr Sh3-Sh2-High Affinity Linker Mutant 3 (Hal3) Domains.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: GOL
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Nef Sf2 Dimerization Mutant Bound To Hck Sh3
Organism: Hiv-1 m:b_arv2/sf2, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-07-15 Classification: VIRAL PROTEIN |
Organism: Hiv-1 m:b_arv2/sf2, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
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Crystal Structure Of Wdr5 In Complex With Triazole-Based Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2025-08-13 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: A1BW7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-13
Ligands: A1BW7
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Crystal Structure Of Wdr5 In Complex With Triazole-Based Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2025-08-13 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: A1BW8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-13
Ligands: A1BW8
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Crystal Structure Of Wdr5 In Complex With Triazole-Based Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2025-08-13 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: A1BW9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-13
Ligands: A1BW9
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Crystal Structure Of Hck In Complex With The Src-Family Kinase Inhibitor A-419259
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-10-09 Classification: TRANSFERASE Ligands: VSE, EDO, DMS, SCN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: VSE, EDO, DMS, SCN
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Nef Sf2 Dimerization Mutant Bound To Hck Sh3
Organism: Hiv-1 m:b_arv2/sf2, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2023-02-22 Classification: VIRAL PROTEIN |
Organism: Hiv-1 m:b_arv2/sf2, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
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Crystal Structure Of Human Fgr Tyrosine Kinase In Complex With A-419259
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2022-12-28 Classification: TRANSFERASE Ligands: GOL, VSE, CL, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: GOL, VSE, CL, PO4
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Crystal Structure Of Human Fgr Tyrosine Kinase In Complex With Tl02-59
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2022-12-28 Classification: TRANSFERASE Ligands: OJL, EDO, GOL, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: OJL, EDO, GOL, PO4
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Discovery Of Potent Orally Bioavailable Wd Repeat Domain 5 (Wdr5) Inhibitors Using A Pharmacophore-Based Optimization
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2022-05-04 Classification: Transcription/Transcription Inhibitor Ligands: MBU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: MBU
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Wdr5 Bound To 2-(3,5-Dimethoxybenzyl)-7-((2-Methyl-1H-Imidazol-1-Yl)Methyl)-5-(1-Methyl-3-(Trifluoromethyl)-1H-Pyrazol-4-Yl)-3,4-Dihydroisoquinolin-1(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-04-27 Classification: Transcription/Transcription Inhibitor Ligands: BEN, M4U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-27
Ligands: BEN, M4U
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Sars-Cov-2 3Clpro In Complex With 2-(Benzotriazol-1-Yl)-N-[4-(1H-Pyrazol-4-Yl)Phenyl]-N-(3-Thienylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, hydrolase/Inhibitor Ligands: Y6A |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: Y6A
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Sars-Cov-2 3Clpro In Complex With N-[4-[[2-(Benzotriazol-1-Yl)Acetyl]-(3-Thienylmethyl)Amino]Phenyl]Cyclopropanecarboxamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: Y6J |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: Y6J
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Sars-Cov-2 3Clpro In Complex With 2-(Benzotriazol-1-Yl)-N-[4-(1H-Imidazol-4-Yl)Phenyl]-N-(3-Thienylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: Y6G |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: Y6G
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Sars-Cov-1 3Clpro In Complex With N-(4-(1H-Imidazol-4-Yl)Phenyl)-2-(1H-Benzo[D][1,2,3]Triazol-1-Yl)-N-(Thiophen-3-Ylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: GOL, Y6G, PEG |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: GOL, Y6G, PEG
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Sars-Cov-1 3Clpro In Complex With 2-(1H-Benzo[D][1,2,3]Triazol-1-Yl)-N-(4-(Pyridin-3-Yl)Phenyl)-N-(Thiophen-3-Ylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: Y6D, GOL |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: Y6D, GOL
