Search Count: 42
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Structure Of Plasmodium Falciparum 20S Proteasome Bound To An Asparagine-Ethylenediamine Based Inhibitor Tdi6245
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY Resolution:2.86 Å Release Date: 2026-07-29 Classification: HYDROLASE Ligands: A1CRS |
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY
Release Date: 2026-07-29
Ligands: A1CRS
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Crystal Structure Of The Plasmodium Falciparum Apical Membrane Antigen (Ama1) In Complex With Single Domain I-Body Wd34
Organism: Plasmodium falciparum 3d7, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2024-07-03 Classification: PROTEIN BINDING Ligands: MPD, EPE, NA |
Organism: Plasmodium falciparum 3d7, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MPD, EPE, NA
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Crystal Structure Of The Plasmodium Vivax Apical Membrane Antigen (Ama1) In Complex With Single Domain I-Body Wd34
Organism: Plasmodium vivax sal-1, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2024-07-03 Classification: PROTEIN BINDING |
Organism: Plasmodium vivax sal-1, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
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Bile Salt Hydrolase A From Lactobacillus Acidophilus
Organism: Lactobacillus acidophilus
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2023-01-25 Classification: HYDROLASE |
Organism: Lactobacillus acidophilus
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
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Bile Salt Hydrolase A From Lactobacillus Gasseri With Taurine Bound
Organism: Lactobacillus gasseri
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2023-01-25 Classification: HYDROLASE Ligands: TAU, K |
Organism: Lactobacillus gasseri
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
Ligands: TAU, K
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Bile Salt Hydrolase A From Lactobacillus Gasseri With Chenodeoxycholate And Taurine Bound
Organism: Lactobacillus gasseri
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2023-01-25 Classification: HYDROLASE Ligands: TAU, JN3 |
Organism: Lactobacillus gasseri
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
Ligands: TAU, JN3
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Bile Salt Hydrolase B From Lactobacillus Gasseri
Organism: Lactobacillus gasseri
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2023-01-25 Classification: HYDROLASE Ligands: MG |
Organism: Lactobacillus gasseri
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
Ligands: MG
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Bile Salt Hydrolase C From Lactobacillus Johnsonii
Organism: Lactobacillus johnsonii
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2023-01-25 Classification: HYDROLASE |
Organism: Lactobacillus johnsonii
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
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Bile Salt Hydrolase From Lactobacillus Ingluviei
Organism: Lactobacillus ingluviei
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2023-01-25 Classification: HYDROLASE Ligands: PG4, PEG, PGE, CA |
Organism: Lactobacillus ingluviei
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
Ligands: PG4, PEG, PGE, CA
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Bile Salt Hydrolase From Lactobacillus Reuteri
Organism: Lactobacillus reuteri
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2023-01-25 Classification: HYDROLASE Ligands: SO4 |
Organism: Lactobacillus reuteri
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
Ligands: SO4
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Human Soluble Adenylyl Cyclase In Complex With The Inhibitor Tdi10229
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-10-06 Classification: SIGNALING PROTEIN Ligands: 1S2, ACT, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 1S2, ACT, DMS, EDO
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Crystal Structure Of Setd2 Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-09-22 Classification: TRANSFERASE Ligands: ZN, SAM, YJ1, BME |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: ZN, SAM, YJ1, BME
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Crystal Structure Of Setd2 Bound To Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-09-22 Classification: TRANSFERASE Ligands: ZN, SAM, YHY, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: ZN, SAM, YHY, EDO, DMS
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Crystal Structure Of Setd2 Bound To Compound 57
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2021-09-22 Classification: TRANSFERASE Ligands: ZN, SAM, YHV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: ZN, SAM, YHV, EDO
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Macrocyclic Peptides Tdi5575 That Selectively Inhibit The Mycobacterium Tuberculosis Proteasome
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-04-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: U5Y, CIT, DMF |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2021-04-28
Ligands: U5Y, CIT, DMF
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Structure Of Mtb Lpd Bound To 010705
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2021-01-27 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: FAD, WPM, GOL |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2021-01-27
Ligands: FAD, WPM, GOL
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor A85
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMF, M6M, CIT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: DMF, M6M, CIT
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor A86
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMF, M6Y, CIT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: DMF, M6Y, CIT
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor B6
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: M9G |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: M9G
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Integrin Alphavbeta3 Ectodomain Bound To Antagonist Tdi-4161
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2019-09-25 Classification: CELL ADHESION Ligands: NAG, MN, JUY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: NAG, MN, JUY
