Search Count: 22
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Structure Guided Optimisation Of Niclosamide Derivatives As Direct Stat3 Inhibitors Targeting A Novel Binding Site
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2026-06-24 Classification: DNA BINDING PROTEIN Ligands: VUT |
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-24
Ligands: VUT
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Crystal Structure Of Beta-Trcp Bound By Diphosphorylated I-Kappa-B-Alpha Degron Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2026-04-08 Classification: TRANSFERASE Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
Ligands: EDO
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Crystal Structure Of Beta-Trcp Bound By Diphosphorylated Claspin Degron Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2026-04-08 Classification: TRANSFERASE Ligands: EDO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
Ligands: EDO, MG
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Crystal Structure Of Beta-Trcp Bound By Diphosphorylated Pdcd4 Degron Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2026-04-08 Classification: TRANSFERASE Ligands: MG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
Ligands: MG, EDO
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Crystal Structure Of Beta-Trcp Bound By Monophosphorylated Atf4 Degron Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-04-08 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
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Crystal Structure Of Beta-Trcp Bound By Monophosphorylated Wee1 Degron Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2026-04-08 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-08
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Keap1 - Inhibitor Complex - 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2026-03-11 Classification: PEPTIDE BINDING PROTEIN Ligands: DMS, A1JB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-11
Ligands: DMS, A1JB1
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Keap1 - Inhibitor Complex - 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2026-03-11 Classification: PEPTIDE BINDING PROTEIN Ligands: A1JBX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-11
Ligands: A1JBX
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Keap1 - Inhibitor Complex - 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2026-03-11 Classification: PEPTIDE BINDING PROTEIN Ligands: A1JB1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-11
Ligands: A1JB1, EDO
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C-Terminal Head Domain Of The Trimeric Autotransporter Adhesin Bpac From Burkholderia Pseudomallei Fused To A Gcn4 Anchor
Organism: Burkholderia pseudomallei 1026b, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2022-06-29 Classification: CELL ADHESION Ligands: GOL, NA |
Organism: Burkholderia pseudomallei 1026b, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2022-06-29
Ligands: GOL, NA
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Crystal Structure Of The Human Mgc45594 Gene Product In Complex With Celecoxib.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2022-05-04 Classification: OXIDOREDUCTASE Ligands: NAP, CEL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: NAP, CEL
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Keap1 - Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2019-10-30 Classification: PEPTIDE BINDING PROTEIN Ligands: EDO, GX8, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-30
Ligands: EDO, GX8, NA
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Crystal Structure Of Spindlin1 In Complex With The Methyltransferase Inhibitor A366
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2018-12-26 Classification: GENE REGULATION Ligands: 2OD, EDO, DMS, MPD, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: 2OD, EDO, DMS, MPD, GOL, NA
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Crystal Structure Of Spindlin1 In Complex With The Inhibitor Vinspinin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2018-12-05 Classification: CELL CYCLE Ligands: H7T, DMS, GLY, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-05
Ligands: H7T, DMS, GLY, PO4
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Crystal Structure Of Spindlin1 In Complex With The Inhibitor Td001851A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2018-12-05 Classification: CELL CYCLE Ligands: MPD, MRD, DMS, H7Q, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-05
Ligands: MPD, MRD, DMS, H7Q, CL
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Keap1 - Peptide Complex
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2018-08-08 Classification: PEPTIDE BINDING PROTEIN Ligands: ACT, EDO, CL, NA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: ACT, EDO, CL, NA
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Keap1 - Peptide Complex
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-08-08 Classification: PEPTIDE BINDING PROTEIN Ligands: EDO, ACT, NA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: EDO, ACT, NA
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Ticagrelor Antidote Candidate Medi2452 In Complex With Ticagrelor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2015-04-01 Classification: IMMUNE SYSTEM Ligands: TIQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-01
Ligands: TIQ
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Ticagrelor Antidote Candidate Fab 72 In Complex With Ticagrelor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-04-01 Classification: IMMUNE SYSTEM Ligands: TIQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-01
Ligands: TIQ
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I45T Cytosolic Phosphoenolpyruvate Carboxykinase In Complex With Beta-Sulfopyruvate And Gtp
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-06-11 Classification: LYASE Ligands: MN, GTP, SPV, NA, 1PE, ETX |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: MN, GTP, SPV, NA, 1PE, ETX
