Search Count: 53
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Crystal Structure Of The Glp (Ehmt1) Set Domain In Complex With Sam And Tng917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2026-05-13 Classification: TRANSFERASE Ligands: ZN, SAM, A1CXM, PEG, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: ZN, SAM, A1CXM, PEG, SO4, EDO
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Crystal Structure Of The G9A (Ehmt2) Set Domain In Complex With Sam And Tng917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2026-05-13 Classification: TRANSFERASE Ligands: ZN, SAM, A1CXM, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: ZN, SAM, A1CXM, EDO, GOL
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Cdk9/Cyclin T1 In Complex With Kb-0742
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.75 Å Release Date: 2023-12-06 Classification: TRANSCRIPTION Ligands: VQE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: VQE
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Crystal Structure Of Human Csnk1A1 With A86
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: DMS, PGE, EDO, PEG, TCE, LCI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: DMS, PGE, EDO, PEG, TCE, LCI
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Crystal Structure Of Human Cdk9/Cyclint1 With A86
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.17 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: LCI, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: LCI, GOL
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Crystal Structure Of Human Ckidelta With A86
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2018-08-29 Classification: TRANSFERASE Ligands: CIT, GOL, LCI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: CIT, GOL, LCI
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Crystal Structure Of Hiv Protease Complexed With Methyl N-[(1S)-1-Benzhydryl-2-(3-Morpholin-4-Ium-2-Ylpropylamino)-2-Oxo-Ethyl]Carbamate
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2016-05-18 Classification: HYDROLASE/INHIBITOR Ligands: 6EH, CL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6EH, CL
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Crystal Structure Of Hiv Protease Complexed With Methyl N-[(1S)-1-[[2-[(3S)-3-[(4-Aminophenyl)Methylamino]-4-Hydroxy-Butyl]Phenyl]Carbamoyl]-2,2-Diphenyl-Ethyl]Carbamate
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-05-18 Classification: HYDROLASE/INHIBITOR Ligands: CL, 6EG |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: CL, 6EG
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Crystal Structure Of Hiv Protease Complexed With Methyl N-[(1S)-1-Benzhydryl-2-[2-[2-[(2R,5S)-5-(Benzylcarbamoyloxymethyl)Morpholin-2-Yl]Ethyl]Anilino]-2-Oxo-Ethyl]Carbamate
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2016-05-18 Classification: HYDROLASE/INHIBITOR Ligands: CL, 6EF |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: CL, 6EF
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Crystal Structure Of Hiv Protease Complexed With [(1S)-1-[(S)-(4-Chlorophenyl)-(3,5-Difluorophenyl)Methyl]-2-[[5-Fluoro-4-[2-[(2R,5S)-5-(2,2,2-Trifluoroethylcarbamoyloxymethyl)Morpholin-4-Ium-2-Yl]Ethyl]Pyridin-1-Ium-3-Yl]Amino]-2-Oxo-Ethyl]Ammonium
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2016-05-18 Classification: HYDROLASE/INHIBITOR Ligands: ACT, 6EE, CL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: ACT, 6EE, CL
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Bace1 In Complex With 4-(Cyclohexylamino)-1-(3-Fluorophenyl)-8-(3-Isopropoxybenzyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QA
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Bace1 In Complex With 8-(3-((1-Aminopropan-2-Yl)Oxy)Benzyl)-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: 4QD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QD
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Bace1 In Complex With 8-Benzyl-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-7-Methyl-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QF
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Discovery Of Doravirine, An Orally Bioavailable Non-Nucleoside Reverse Transcriptase Inhibitor Potent Against A Wide Range Of Resistant Mutant Hiv Viruses
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-02-12 Classification: Transferase/Inhhibitor, Hydrolase/Inhhibitor Ligands: 2KW |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: 2KW
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Discovery Of Pyrrolidine-Based B-Secretase Inhibitors: Lead Advancement Through Conformational Design For Maintenance Of Ligand Binding Efficiency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-01-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 508, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
Ligands: 508, SO4, GOL
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Crystal Structure Of Hiv-1 Reverse Transcriptase (Wild Type) In Complex With Inhibitor M05
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-10-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5MA |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: 5MA
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Crystal Structure Of Hiv-1 Reverse Transcriptase (K103N Mutant) In Complex With Inhibitor M05
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2011-10-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5MA |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: 5MA
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Crystal Structure Of Hiv-1 Reverse Transcriptase (K103N Mutant) In Complex With Inhibitor M06
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2011-10-26 Classification: Transferase/transferase Inhibitor Ligands: M06 |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: M06
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Hiv Protease Complexed With Compound 10B
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-06-30 Classification: TRANSFERASE Ligands: 595, CL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2010-06-30
Ligands: 595, CL
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Crystal Structure Of Hiv Reverse Transcriptase In Complex With Inhibitor 3
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2009-08-25 Classification: TRANSFERASE Ligands: RT3 |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: RT3