Search Count: 22
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Pkr Kinase Domain - Dabrafenib Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-07-01 Classification: TRANSFERASE/INHIBITOR Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: P06
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Crystal Structure Of Dcaf1 In Complex With Sdiptac C11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2026-06-10 Classification: PROTEIN BINDING Ligands: A1C24, A1C27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1C24, A1C27
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Crystal Structure Of Dcaf1 In Complex With Sdiptac C7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2026-05-20 Classification: PROTEIN BINDING Ligands: A1C24, A1C23 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-20
Ligands: A1C24, A1C23
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Crystal Structure Of Dcaf1 In Complex With Sdiptac C8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2026-05-20 Classification: PROTEIN BINDING Ligands: A1C24, A1C25 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-20
Ligands: A1C24, A1C25
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Crystal Structure Of Dcaf1 In Complex With Sdiptac C9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-05-20 Classification: PROTEIN BINDING Ligands: A1C24, A1C26 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-20
Ligands: A1C24, A1C26
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Crystal Structure Of The Human Dcaf1 Wdr Domain In Complex With Oicr-41109
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-11-26 Classification: TRANSPORT PROTEIN Ligands: A1CY9, NA, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-26
Ligands: A1CY9, NA, UNX
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Crystal Structure Of The Ternary Complex Of Dcaf1 And Wdr5 With Protac, Oicr-40333
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2024-11-06 Classification: PROTEIN BINDING Ligands: A1AM2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1AM2
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Crystal Structure Of The Ternary Complex Of Dcaf1 And Wdr5 With Protac, Oicr-40407
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2024-11-06 Classification: PROTEIN BINDING Ligands: A1ANM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ANM
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Crystal Structure Of The Ternary Complex Of Dcaf1 And Wdr5 With Protac, Oicr-40792
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2024-11-06 Classification: PROTEIN BINDING Ligands: A1ANN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1ANN
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Crystal Structure Of The Binary Complex Of Dcaf1 And Wdr5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.97 Å Release Date: 2024-11-06 Classification: PROTEIN BINDING Ligands: IMD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: IMD
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Crystal Structure Of The Ternary Complex Of Dcaf1 And Wdr5 With Protac, Oicr-41114
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-11-06 Classification: PROTEIN BINDING Ligands: A1BAF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1BAF
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Oicr-4425
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2022-08-17 Classification: TRANSCRIPTION/INHIBITOR Ligands: YJV, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: YJV, DMS
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Oicr-11029
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2022-03-16 Classification: TRANSCRIPTION/INHIBITOR Ligands: YJS, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: YJS, DMS, SO4
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Oicr-7629
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.17 Å Release Date: 2022-03-09 Classification: TRANSCRIPTION/INHIBITOR Ligands: YND, FMT, ACT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-09
Ligands: YND, FMT, ACT, CL
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Oicr-9320
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2022-03-09 Classification: TRANSCRIPTION/INHIBITOR Ligands: YNA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-09
Ligands: YNA, GOL
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Oicr-12694
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2022-03-09 Classification: TRANSCRIPTION/INHIBITOR Ligands: YN7, GOL, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-09
Ligands: YN7, GOL, UNX
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Crystal Structure Of Braf Kinase Domain Bound To The Protac P4B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.29 Å Release Date: 2020-06-03 Classification: SIGNALING PROTEIN Ligands: QH1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: QH1
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Crystal Structure Of The Acvr1 (Alk2) Kinase In Complex With The Compound M4K2009
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2019-10-16 Classification: SIGNALING PROTEIN Ligands: M2Z, SO4, EDO, NH4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-16
Ligands: M2Z, SO4, EDO, NH4, DMS
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Crystal Structure Of Murine Ire1 In Complex With Mkc9989 Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-09-03 Classification: TRANSFERASE,HYDROLASE/INHIBITOR Ligands: 31J, ADP, MG |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 31J, ADP, MG
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Crystal Structure Of Murine Ire1 In Complex With Oicr464 Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2014-09-03 Classification: TRANSFERASE,HYDROLASE/INHIBITOR Ligands: 31K, ADP, PEU, MG |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 31K, ADP, PEU, MG
