Search Count: 28
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Human Rock2 In Complex With A Dihydropyrazolo-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2026-06-10 Classification: TRANSFERASE Ligands: A1I40 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1I40
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Structure Of An Inhibitor Of Human Tgf-Beta Type I Receptor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2026-05-27 Classification: TRANSFERASE Ligands: A1JQO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1JQO, GOL
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Human Pi3Kdelta In Complex With Isocumarin Inhibitor Chf-6523
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1IJ5 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1IJ5
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Human Pi3Kdelta In Complex With Isocumarin Inhibitor 10
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1IJ1, CL |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1IJ1, CL
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Human Pi3Kgamma In Complex With Isocumarin Inhibitor 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1IKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1IKW, SO4
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Crystal Structure Of Rock2 In Complex With A 8-(Azaindolyl)-Benzoazepinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2024-09-25 Classification: TRANSFERASE Ligands: A1H6L, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-25
Ligands: A1H6L, EDO
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E.Coli Yihx Wild Type Apo
Organism: Escherichia coli str. k-12 substr. mg1655
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-07-10 Classification: HYDROLASE Ligands: PEG, GOL, MG, CA, CL |
Organism: Escherichia coli str. k-12 substr. mg1655
Method: X-RAY DIFFRACTION
Release Date: 2024-07-10
Ligands: PEG, GOL, MG, CA, CL
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The Mgf3(H2O) Transition State Analog Complex Of E. Coli Yihx
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2024-07-10 Classification: HYDROLASE Ligands: PEG, KQB, PG4, IMD, EDO, MG, GOL, CA |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2024-07-10
Ligands: PEG, KQB, PG4, IMD, EDO, MG, GOL, CA
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Human Pi3Kdelta In Complex With Pyridazinone Inhibitor 7
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2024-07-03 Classification: TRANSFERASE Ligands: A1H48 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: A1H48
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Oxa-48 With Carbamylated Lys73 In Complex With Hydrolysed Imipenem And Bromide Ion Competing For Binding With Arg250 At Neutral Ph
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2023-11-08 Classification: HYDROLASE Ligands: 8YF, BR, 1BO |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: 8YF, BR, 1BO
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Human Pi3Kdelta In Complex With Compound 13
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2023-05-10 Classification: TRANSFERASE Ligands: I3H |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2023-05-10
Ligands: I3H
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Acetyllysine73-Incorporated Oxa-48 Complexed With Imipenem And Bromide Ions In Both Active And Inactive Acyl-Enzyme Intermediates
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-11-16 Classification: HYDROLASE Ligands: ID1, 1BO, BR |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-11-16
Ligands: ID1, 1BO, BR
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Acetyllysine73-Incorporated Oxa-48 Complexed With Oxacillin
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2022-10-05 Classification: HYDROLASE Ligands: 1S6, 1BO, CL |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: 1S6, 1BO, CL
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Crystal Structure Of A Class D Carbapenemase Complexed With Imipenem
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-10-05 Classification: HYDROLASE Ligands: ID1, BR, 1BO |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: ID1, BR, 1BO
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Apo Oxa-48 With Fully Carbamylated Lys73 At Ph 7.5
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2022-08-24 Classification: HYDROLASE Ligands: 1BO |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 1BO
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Oxa-48_E185A/R186A/R206A With Carbamylated Lys73 In Complex With Chloride Ions At Neutral Ph
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-08-24 Classification: HYDROLASE Ligands: GOL, SO4 |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: GOL, SO4
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Crystal Structure Of A Class D Carbapenemase Complexed With Hydrolyzed Imipenem
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-08-24 Classification: HYDROLASE Ligands: HIW, BR, 1BO |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: HIW, BR, 1BO
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Acetyllysine73-Incorporated Oxa-48 Complexed With Imipenem In Both Active And Inactive Acyl-Enzyme Intermediates
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-08-24 Classification: HYDROLASE Ligands: ID1, 1BO, PO4 |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: ID1, 1BO, PO4
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Oxa-48_R250A With Carbamylated Lys73 With Bromide Ions Bound At Neutral Ph
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2022-08-24 Classification: HYDROLASE Ligands: 1BO, BR |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 1BO, BR
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Oxa-48 With Carbamylated Lys73 In Complex With Bicarbonate Ions At Neutral Ph
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-05-04 Classification: HYDROLASE Ligands: BCT |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: BCT
