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9Y0G image
Crystal Structure Of Nras-G12D In Complex With Gdp And Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2026-02-25
Classification: HYDROLASE
Ligands: GDP, A1CRR, MG, CIT

9Y1W image
Crystal Structure Of Nras-G12D In Complex With Gdp And Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2026-02-25
Classification: HYDROLASE
Ligands: GDP, MG, A1CRV, CIT

9Y1X image
Crystal Structure Of Nras-G12D In Complex With Gdp And Iacs-56676
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2026-02-25
Classification: HYDROLASE
Ligands: GDP, A1CRW, MG, CIT

9Y1Y image
Crystal Structure Of Nras-G12D In Complex With Gdp And Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2026-02-25
Classification: HYDROLASE
Ligands: GDP, MG, A1CR1, CIT

9Y1Z image
Crystal Structure Of Nras-G12D In Complex With Gdp And Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.92 Å Release Date: 2026-02-25
Classification: HYDROLASE
Ligands: GDP, MG, A1CR2, CIT

9Y3W image
Crystal Structure Of Nras-G12D In Complex With Gdp And Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.56 Å Release Date: 2026-02-25
Classification: HYDROLASE
Ligands: GDP, MG, A1CSD, CIT

9HDF image
Glucocorticoid Receptor Ligand Binding Domain In Complex With Dexamethasone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.78 Å Release Date: 2025-11-12
Classification: DNA BINDING PROTEIN
Ligands: DEX, CAC, EPE, GOL, SO4, CL, PG4, IMD, PEG, PGE

9GC4 image
Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.42 Å Release Date: 2025-02-12
Classification: SIGNALING PROTEIN
Ligands: A1IZ7

9GC5 image
Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.91 Å Release Date: 2025-02-12
Classification: SIGNALING PROTEIN
Ligands: A1IZ8, SO4

9GC6 image
Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2025-02-12
Classification: SIGNALING PROTEIN
Ligands: A1IZ9

9GDV image
Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.22 Å Release Date: 2025-02-12
Classification: SIGNALING PROTEIN
Ligands: Q6K, SO4

9HBO image
Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations. Compound 51 Bound To Egfrinsnpg [V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.45 Å Release Date: 2025-02-05
Classification: SIGNALING PROTEIN
Ligands: A1IUK

8V5H image
Crystal Structure Of Mastl Kinase Domain In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.74 Å Release Date: 2025-01-22
Classification: TRANSFERASE/INHIBITOR
Ligands: A1AAE

8V5I image
Crystal Structure Of Map4K4 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.18 Å Release Date: 2025-01-22
Classification: TRANSFERASE/INHIBITOR
Ligands: A1AAA

9CZT image
Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.69 Å Release Date: 2024-12-18
Classification: TRANSFERASE
Ligands: A1A1E

9CZU image
Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2024-12-18
Classification: TRANSFERASE
Ligands: SO4, A1A1D

9CZW image
Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.59 Å Release Date: 2024-12-18
Classification: TRANSFERASE
Ligands: A1A1C

9CZX image
Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.46 Å Release Date: 2024-12-18
Classification: TRANSFERASE
Ligands: A1A1B, CL

9D00 image
Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2024-12-18
Classification: TRANSFERASE
Ligands: A1A1A

8CDW image
Crystal Structure Of Human Hpk1 (Map4K1) Complex With 7-(1-Methyl-1H-Pyrazol-4-Yl)-N-[4-(1-Methylpiperidin-4-Yl)Phenyl]Quinazolin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.94 Å Release Date: 2023-08-16
Classification: TRANSFERASE
Ligands: UES
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