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Crystal Structure Of Epoxomicin:20S Proteasome Reveals A Molecular Basis For Selectivity Of Alpha,Beta-Epoxyketone Proteasome Inhibitors
Organism: Saccharomyces cerevisiae, Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2000-11-27 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: MG |
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Organism: Bifidobacterium longum
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2023-11-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: WSR |
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Room Temperature X-Ray Structure Of Sars Cov-2 Main Protease Intermediate Precursor With Ensitrelvir (Esv)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2026-05-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7YY |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z2697514548
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: GWG |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With En300-1605072
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: ZQG |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z319891284
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, ZQD |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z2856434783
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: O3G |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z239136710
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: K3A |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z1673618163
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: WL7 |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z59181945
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, VWG |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z31504642
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, WJD |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With En300-321461
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, WOY |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z425449682
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: EJW |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z1530301542
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CIT, ZQA |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With Z68299550
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: JOV |
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Pandda Analysis Group Deposition -- Crystal Structure Of Sars-Cov-2 Nendou In Complex With En300-100112
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2021-06-09 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: ZQJ |
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Organism: Bifidobacterium longum
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-11-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: WU5 |
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Bile Salt Hydrolase B From Lactobacillus Gasseri With Covalent Inhibitor Bound
Organism: Lactobacillus gasseri
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2023-11-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: WU5, NI |
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Human Liver Fructose-1,6-Bisphosphatase(D-Fructose-1,6-Bisphosphate, 1-Phosphohydrolase) (E.C.3.1.3.11) Complexed With The Allosteric Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-11-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2C1 |
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Joint X-Ray/Neutron Structure Of Hiv-1 Protease Triple Mutant (V32I,I47V,V82I) With Darunavir At Ph 4.3
Organism: Human immunodeficiency virus type 1 group m subtype b
Method: X-RAY DIFFRACTION, NEUTRON DIFFRACTION Resolution:1.75 Å, 2.30 Å Release Date: 2016-05-04 Classification: Hydrolase/hydrolase inhibitor Ligands: 017, DOD |




















