Search Count: 23
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Kat6A In Complex With Small Molecule Inhibitor Bay-184
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2024-11-06 Classification: TRANSFERASE Ligands: ZN, A1IDR, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: ZN, A1IDR, EPE
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X-Ray Structure Of Smyd3 In Complex With Benzodiazepine-Type Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZT, SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZT, SAM, ZN
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X-Ray Structure Of Smyd3 In Complex With Benzodiazepine-Type Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZQ, ZN, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZQ, ZN, SAM
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X-Ray Structure Of Smyd3 In Complex With The Benzodiazepine-Based Probe Bay-6035
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: UZK, SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: UZK, SAM, ZN
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X-Ray Structure Of Human K-Ras G12C In Complex With Covalent Isoquinolinone Inhibitor (Compound 3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2020-04-08 Classification: HYDROLASE Ligands: GDP, MG, MZQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GDP, MG, MZQ
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X-Ray Structure Of Human K-Ras G12C In Complex With Covalent Isoquinolinone Inhibitor (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2020-04-08 Classification: HYDROLASE Ligands: GDP, MG, MZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GDP, MG, MZN
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Human Gpx4 In Complex With Covalent Inhibitor Ml162 (S Enantiomer)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2020-04-01 Classification: OXIDOREDUCTASE Ligands: G9N, SO4, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: G9N, SO4, EDO, DMS
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Wildtype Form (Apo) Of Human Gpx4 With Se-Cys46
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2020-04-01 Classification: OXIDOREDUCTASE Ligands: CL, EOH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: CL, EOH, GOL
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Tbk1 In Complex With Inhibitor Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2020-04-01 Classification: IMMUNE SYSTEM Ligands: KJB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: KJB
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Tbk1 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2020-01-01 Classification: IMMUNE SYSTEM Ligands: KHT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: KHT
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Tbk1 In Complex With Inhibitor Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.29 Å Release Date: 2020-01-01 Classification: IMMUNE SYSTEM Ligands: KHQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: KHQ
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Crystal Structure Of Human Dhodh In Complex With Bay 2402234
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2019-06-05 Classification: OXIDOREDUCTASE Ligands: ORO, FMN, JJE, SO4, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-05
Ligands: ORO, FMN, JJE, SO4, ACT
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Jak2 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-[(8As)-2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(8Ah)-Yl]Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
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Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
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Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor (Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexyl)Acetonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J6
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 15T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 15T
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B-Raf Kinase Domain In Complex With An Aminothienopyrimidine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI8
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B-Raf Kinase Domain In Complex With An Aminopyridimine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: RI9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: RI9
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The Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2012-07-04 Classification: Transferase/Transferase Inhibitor Ligands: JAK, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: JAK, EDO
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: 0Q2
