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Cryo-Em Structure Of Ternary Complex Bcl6-Crbn-Ddb1 With Bms-986458 (Local Refined), A Potent And Selective Bcl6 Ligand Directed Degrader (Ldd)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.09 Å Release Date: 2026-02-18 Classification: LIGASE Ligands: A1CTU, ZN |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2026-01-14 Classification: TRANSCRIPTION Ligands: A1CNQ |
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.20 Å Release Date: 2026-01-14 Classification: LIGASE Ligands: ZN, A1CN1 |
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-10-15 Classification: LIGASE Ligands: ZN, A1AF4 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2021-03-24 Classification: LIGASE/LIGASE inhibitor Ligands: SO4, ZN, VB7 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-03-24 Classification: LIGASE/LIGASE inhibitor Ligands: SO4, ZN, VBA |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-10 Classification: LIGASE/LIGASE inhibitor Ligands: SO4, ZN, VAY |
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Monophosphorylated Pser33 B-Catenin Peptide, B-Trcp/Skp1, Nrx-2776 Ternary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: J91, PO4 |
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Monophosphorylated Pser33 B-Catenin Peptide, B-Trcp/Skp1, Nrx-103094 Ternary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: J97, PO4, CL |
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Monophosphorylated Pser33 B-Catenin Peptide, B-Trcp/Skp1, Nrx-2663 Ternary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: J8V, PO4 |
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Monophosphorylated Pser33 B-Catenin Peptide, B-Trcp/Skp1, Nrx-1933 Ternary Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: J8Y, PO4 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-04-03 Classification: LIGASE Ligands: PO4, DMS |
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Structure Of Ubiquitin Activating Enzyme (Uba1) In Complex With Ubiquitin And Tak-243
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-11-01 Classification: LIGASE/LIGASE INHIBITOR Ligands: 61T |













