Search Count: 28
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Cryo-Em Structure Of Ternary Complex Bcl6-Crbn-Ddb1 With Bms-986458 (Local Refined), A Potent And Selective Bcl6 Ligand Directed Degrader (Ldd)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.09 Å Release Date: 2026-02-18 Classification: LIGASE Ligands: A1CTU, ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-02-18
Ligands: A1CTU, ZN
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Blimp-1 With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2026-01-14 Classification: TRANSCRIPTION Ligands: A1CNQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-14
Ligands: A1CNQ
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Cereblon Ternary Complex With Blimp1 And Compound 5
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.20 Å Release Date: 2026-01-14 Classification: LIGASE Ligands: ZN, A1CN1 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-01-14
Ligands: ZN, A1CN1
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Cryo-Em Structure Of Ternary Complex Bcl6-Crbn-Ddb1 With Bcl6-760 (Ldd, Local Refined)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.15 Å Release Date: 2025-10-15 Classification: LIGASE Ligands: ZN, A1CM7 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-10-15
Ligands: ZN, A1CM7
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Crystal Structure Of Ternary Complex Helios-Zf2:I-19:Crbn:Ddb1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.41 Å Release Date: 2025-10-01 Classification: LIGASE Ligands: A1CNP, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-01
Ligands: A1CNP, ZN
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Cryo-Em Structure Of Ternary Complex Ikaros-Zf2:Cc-885:Crbn:Ddb1 (Molecular Glue Degrader)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:2.94 Å Release Date: 2025-10-01 Classification: LIGASE Ligands: ZN, 85C |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-10-01
Ligands: ZN, 85C
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Monkey Tlr7 Ectodomain With Small Molecule Agonist 9
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, CL, A1BLT, CIT |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: NAG, CL, A1BLT, CIT
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Human Tlr8 Ectodomain With Small Molecule Agonist 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, NI, A1BLT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: NAG, NI, A1BLT
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Human Tlr8 Ectodomain With Small Molecule Agonist 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, A1BLO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: NAG, A1BLO
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Human Tlr8 Ectodomain With Small Molecule Agonist 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, SO4, A1BLN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: NAG, SO4, A1BLN
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Cryo-Em Structure Of Human Cereblon/Ddb1 In Complex With A Non-Traditional Crbn Binder
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-12-25 Classification: LIGASE Ligands: ZN, A1BEP |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-12-25
Ligands: ZN, A1BEP
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Crystal Structure Of Mouse Btk Kinase Domain In Complex With Compound 9A
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-01-30 Classification: TRANSFERASE Ligands: JVP |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-01-30
Ligands: JVP
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Human Retenoid-Related Orphan Receptor-Gamma Ligand- Binding Domain In Complex With Indole Ligand Cp9B In Inverse Agonist Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-09-05 Classification: SIGNALING PROTEIN Ligands: F7M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: F7M
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Rorc2 Lbd Complexed With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-09-05 Classification: SIGNALING PROTEIN Ligands: F7J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: F7J
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Crystal Structure Of Ask1 Kinase Domain With A Potent Inhibitor (Analog 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2018-01-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 9E1, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: 9E1, DMS
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Crystal Structure Of Ask1 Kinase Domain With A Potent Inhibitor (Analog 13)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2018-01-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 9E4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: 9E4
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Crystal Structure Of Irak4 In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8BV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8BV
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Crystal Structure Of Irak4 In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8BY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8BY
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Crystal Structure Of Irak4 In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8C1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8C1
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Crystal Structure Of Irak4 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8CD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8CD
