Search Count: 7
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Structure Of Plasmodium Falciparum 20S Proteasome Bound To An Asparagine-Ethylenediamine Based Inhibitor Tdi6245
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY Resolution:2.86 Å Release Date: 2026-07-29 Classification: HYDROLASE Ligands: A1CRS |
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY
Release Date: 2026-07-29
Ligands: A1CRS
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Macrocyclic Peptides Tdi5575 That Selectively Inhibit The Mycobacterium Tuberculosis Proteasome
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-04-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: U5Y, CIT, DMF |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2021-04-28
Ligands: U5Y, CIT, DMF
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Structure Of Rorgt In Complex With A Novel Inverse Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2019-07-17 Classification: nuclear protein/agonist Ligands: SO4, MPD, HQ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: SO4, MPD, HQ7
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Structure Of Rorgt In Complex With A Novel Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-06-12 Classification: nuclear protein/agonist Ligands: EDO, HOJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: EDO, HOJ
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Structure Of Rorgt In Complex With A Novel Isoquinoline Inverse Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2018-03-21 Classification: transcription/agonist Ligands: MPD, E3S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: MPD, E3S
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Structure Of Rorgt In Complex With A Novel Inverse Agonist Tak-828.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2018-03-21 Classification: transcription/agonist Ligands: MPD, E3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: MPD, E3V
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Structure Of Protein Kinase C Theta With Compound 10: 2,2-Dimethyl-7-(2-Oxidanylidene-3~{H}-Imidazo[4,5-B]Pyridin-1-Yl)-1-(Phenylmethyl)-3~{H}-Quinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-05-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5VS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-11
Ligands: 5VS
