Search Count: 24
![]() |
Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn012042
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: XRM, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: XRM, CL, EDO
![]() |
Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn011980
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: YFG, CL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: YFG, CL, GOL
![]() |
Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn012759
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2021-03-24 Classification: TRANSFERASE/Inhibitor Ligands: XBA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: XBA, EDO
![]() |
Human Parp14 (Artd8), Catalytic Fragment In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2021-03-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: TZ7, EDO, PEG, GOL, SO4, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: TZ7, EDO, PEG, GOL, SO4, PGE
![]() |
Human Parp14 (Artd8), Catalytic Fragment In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2021-03-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: FDR, EDO, TYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: FDR, EDO, TYG, GOL
![]() |
Human Poly(Adp-Ribose) Polymerase 12, Catalytic Fragment With Four Point Mutations In Complex With Rbn-2397
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-12-16 Classification: TRANSFERASE Ligands: QO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: QO4, CL
![]() |
Human Parp16 In Complex With Rbn010860
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2020-10-07 Classification: TRANSFERASE Ligands: T9D, CIT, GOL, EDO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: T9D, CIT, GOL, EDO, PEG
![]() |
Crystal Structure Of Whsc1L1 In Complex With Inhibitor Pep21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2018-05-09 Classification: TRANSFERASE/INHIBITOR Ligands: SAM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: SAM, ZN
![]() |
Crystal Structure Of Smyd2 With Sam And Epz033294
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-04-25 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SAM, ZN, 8WG, PEG, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-25
Ligands: SAM, ZN, 8WG, PEG, EDO, GOL
![]() |
Crystal Structure Of Smyd3 With Sam And Epz028862
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2018-03-07 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: ZN, SAM, 8WD, PEG, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: ZN, SAM, 8WD, PEG, DMS, EDO
![]() |
Crystal Structure Of Smyd3 With Sam And Oxindole Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2015-09-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, SAM, 4ZW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: ZN, SAM, 4ZW, EDO
![]() |
Crystal Structure Of Smyd3 With Sam And Epz030456
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-09-09 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ZN, SAM, 4ZX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: ZN, SAM, 4ZX
![]() |
Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SFG, 3XV, GOL
![]() |
Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAM, 3XV, GOL
![]() |
Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAH, 3XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 3XV
![]() |
Crystal Structure Of Human Protein Arginine Methyltransferase Prmt6 Bound To Sah And An Aryl Pyrazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: SAH, 49K, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 49K, GOL
![]() |
Crystal Structure Of Human Protein Arginine Methyltransferase Prmt6 Bound To Sah And Epz020411
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-04-22 Classification: TRANSFERASE Ligands: SAH, 49L, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 49L, MG, GOL
![]() |
Crystal Structure Of Human Kdm4C Catalytic Domain With Oga
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2015-03-25 Classification: OXIDOREDUCTASE Ligands: ZN, FE, OGA, PGE, EDO, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: ZN, FE, OGA, PGE, EDO, PG4
![]() |
Crystal Structure Of Human Kdm4C Catalytic Domain Bound To Tris
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2015-03-25 Classification: OXIDOREDUCTASE Ligands: ZN, FE, TRS, PGE, EDO, CL, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: ZN, FE, TRS, PGE, EDO, CL, PG4
![]() |
Crystal Structure Of Dot1L In Complex With Epz000004
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-10-17 Classification: transferase/transferase inhibitor Ligands: EP4, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-17
Ligands: EP4, SO4, GOL
