Search Count: 45
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Crystal Structure Of The Glp (Ehmt1) Set Domain In Complex With Sam And Tng917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2026-05-13 Classification: TRANSFERASE Ligands: ZN, SAM, A1CXM, PEG, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: ZN, SAM, A1CXM, PEG, SO4, EDO
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Crystal Structure Of The G9A (Ehmt2) Set Domain In Complex With Sam And Tng917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2026-05-13 Classification: TRANSFERASE Ligands: ZN, SAM, A1CXM, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-13
Ligands: ZN, SAM, A1CXM, EDO, GOL
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Cdk9/Cyclin T1 In Complex With Kb-0742
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.75 Å Release Date: 2023-12-06 Classification: TRANSCRIPTION Ligands: VQE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: VQE
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Crystal Structure Of Hiv Protease Complexed With Methyl N-[(1S)-1-Benzhydryl-2-(3-Morpholin-4-Ium-2-Ylpropylamino)-2-Oxo-Ethyl]Carbamate
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2016-05-18 Classification: HYDROLASE/INHIBITOR Ligands: 6EH, CL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6EH, CL
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Crystal Structure Of Hiv Protease Complexed With Methyl N-[(1S)-1-[[2-[(3S)-3-[(4-Aminophenyl)Methylamino]-4-Hydroxy-Butyl]Phenyl]Carbamoyl]-2,2-Diphenyl-Ethyl]Carbamate
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-05-18 Classification: HYDROLASE/INHIBITOR Ligands: CL, 6EG |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: CL, 6EG
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Crystal Structure Of Hiv Protease Complexed With Methyl N-[(1S)-1-Benzhydryl-2-[2-[2-[(2R,5S)-5-(Benzylcarbamoyloxymethyl)Morpholin-2-Yl]Ethyl]Anilino]-2-Oxo-Ethyl]Carbamate
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2016-05-18 Classification: HYDROLASE/INHIBITOR Ligands: CL, 6EF |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: CL, 6EF
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Crystal Structure Of Hiv Protease Complexed With [(1S)-1-[(S)-(4-Chlorophenyl)-(3,5-Difluorophenyl)Methyl]-2-[[5-Fluoro-4-[2-[(2R,5S)-5-(2,2,2-Trifluoroethylcarbamoyloxymethyl)Morpholin-4-Ium-2-Yl]Ethyl]Pyridin-1-Ium-3-Yl]Amino]-2-Oxo-Ethyl]Ammonium
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2016-05-18 Classification: HYDROLASE/INHIBITOR Ligands: ACT, 6EE, CL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: ACT, 6EE, CL
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Discovery Of Pyrrolidine-Based B-Secretase Inhibitors: Lead Advancement Through Conformational Design For Maintenance Of Ligand Binding Efficiency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-01-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 508, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
Ligands: 508, SO4, GOL
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Crystal Structure Of Hiv-1 Reverse Transcriptase (Wild Type) In Complex With Inhibitor M05
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-10-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5MA |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: 5MA
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Crystal Structure Of Hiv-1 Reverse Transcriptase (K103N Mutant) In Complex With Inhibitor M05
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2011-10-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5MA |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: 5MA
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Hiv Protease Complexed With Compound 10B
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-06-30 Classification: TRANSFERASE Ligands: 595, CL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2010-06-30
Ligands: 595, CL
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Crystal Structure Of Hiv Reverse Transcriptase In Complex With Inhibitor 3
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2009-08-25 Classification: TRANSFERASE Ligands: RT3 |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: RT3
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Crystal Structure Of Hiv Reverse Transcriptase In Complex With Inhibitor 7
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-08-25 Classification: TRANSFERASE Ligands: RT7 |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: RT7
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Discovery Of Aminoheterocycles As A Novel Beta-Secretase Inhibitor Class
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: B35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: B35
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Crystal Structure Of Human Beta Secretase Complexed With Spiropiperdine Iminohydantoin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: SII |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: SII
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Hiv Reverse Transcriptase In Complex With Inhibitor R8E
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-10-14 Classification: TRANSFERASE Ligands: R8E |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: R8E
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Hiv Reverse Transcriptase Y181C Mutant In Complex With Inhibitor R8E
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2008-10-14 Classification: TRANSFERASE Ligands: R8E |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: R8E
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Hiv Reverse Transcriptase K103N Mutant In Complex With Inhibitor R8D
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2008-10-14 Classification: TRANSFERASE Ligands: R8D |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: R8D
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Crystal Structure Of Hiv-1 Protease Complexed With Pl-100
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-07-22 Classification: HYDROLASE Ligands: A00 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2008-07-22
Ligands: A00
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Crystal Structure Of Human Beta Secretase Complexed With I21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-04-29 Classification: HYDROLASE Ligands: I21 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-29
Ligands: I21
