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8QDG image
Compound 1A Bound Kmt9 Crystal Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.39 Å Release Date: 2024-09-11
Classification: TRANSFERASE
Ligands: SDU

8QDI image
Compound 1B Bound Kmt9 Crystal Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.47 Å Release Date: 2024-09-11
Classification: TRANSFERASE
Ligands: QII

7PJM image
Crystal Structure Of Ivosidenib-Resistant Idh1 Variant R132C S280F In Complex With Nadph And Ca2+/2-Oxoglutarate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2022-07-13
Classification: OXIDOREDUCTASE
Ligands: AKG, GOL, NDP, CA, CL

7PJN image
Crystal Structure Of Ivosidenib-Resistant Idh1 Variant R132C S280F In Complex With Nadph And Inhibitor Ds-1001B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.45 Å Release Date: 2022-07-13
Classification: OXIDOREDUCTASE
Ligands: 7SU, CIT, GOL, NDP
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