Search Count: 13
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P53-R282W Core Domain Covalently Bound To A Vinyl-Sulfone Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2026-05-27 Classification: CELL CYCLE Ligands: EPE, PEG, A1JQW, GOL, EDO, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: EPE, PEG, A1JQW, GOL, EDO, ZN
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P53-Y220C Core Domain Covalently Bound To A Vinyl-Sulfone Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-05-27 Classification: CELL CYCLE Ligands: A1JQW, EPE, ZN, PGE, PEG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1JQW, EPE, ZN, PGE, PEG, EDO
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Usp7 Covalently Bound To N-(6-Fluoro-3-Nitropyridin-2-Yl)-5-(1-Methyl-1H-Pyrazol-4-Yl)Isoquinolin-3-Amine (Gcl36, 7A) With Partial Occupancy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2025-09-10 Classification: HYDROLASE Ligands: A1I71, EDO, PEG, BR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1I71, EDO, PEG, BR
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P53-Y220C Core Domain Covalently Bound To 2-Chloro-5-Cyanopyrazine Soaked At 5 Mm
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2025-06-11 Classification: CELL CYCLE Ligands: A1IIO, EPE, PEG, EDO, ZN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: A1IIO, EPE, PEG, EDO, ZN, GOL
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P53-Y220C Core Domain Covalently Bound To 5-Chloro-6-Methylpyrazine-2-Carbonitrile Soaked At 5 Mm
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2025-06-11 Classification: CELL CYCLE Ligands: A1II4, EDO, EPE, PEG, GOL, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: A1II4, EDO, EPE, PEG, GOL, ZN
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P53-Y220C Core Domain Covalently Bound To 3,5-Dichloro-6-Ethylpyrazine-2-Carbonitirle Soaked At 5 Mm
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2025-06-11 Classification: CELL CYCLE Ligands: A1II1, PEG, EDO, EPE, ZN, GOL, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: A1II1, PEG, EDO, EPE, ZN, GOL, PGE
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P53-Y220C Core Domain Covalently Bound To 2,5,6-Trifluoropyridine-3-Carbonitrile Soaked At 5 Mm
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2024-11-27 Classification: CELL CYCLE Ligands: YLW, PEG, EDO, EPE, ZN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: YLW, PEG, EDO, EPE, ZN, GOL
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P53-Y220C Core Domain Covalently Bound To 2,5,6-Trifluoropyridine-3-Carbonitrile Soaked At 40 Mm
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2024-11-27 Classification: CELL CYCLE Ligands: YLW, GOL, EDO, EPE, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: YLW, GOL, EDO, EPE, ZN
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P53-Y220C Core Domain Covalently Bound To 3-Amino-5-Chloropyrazine-2,6-Dicarbonitrile Soaked At 5 Mm
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2024-11-27 Classification: CELL CYCLE Ligands: YM0, EPE, PEG, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: YM0, EPE, PEG, ZN
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Dyrk1A In Complex With 2-Cyclopentyl-7-Iodo-1H-Indole-3-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2024-09-25 Classification: TRANSFERASE Ligands: YOX, 1PE, PG4, EPE, PEG, GOL, EDO, SO4, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-25
Ligands: YOX, 1PE, PG4, EPE, PEG, GOL, EDO, SO4, PO4
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Jnk3 (Mitogen-Activated Protein Kinase 10) In Complex With Compound 23 Bearing A C(Sp3)F2Br Moiety
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2023-08-02 Classification: TRANSFERASE Ligands: SWM, EDO, GOL, BME, PEG, C15, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-02
Ligands: SWM, EDO, GOL, BME, PEG, C15, CL
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Dyrk1A In Complex With A Bromo-Triazolo-Pyridine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-11-09 Classification: TRANSFERASE Ligands: IWU, PG4, PEG, PGE, GOL, EPE, 1PE, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: IWU, PG4, PEG, PGE, GOL, EPE, 1PE, SO4, CL
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P53-Y220C Core Domain In Complex With A Bromo-Trifluoro-Pyrazole-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2022-11-09 Classification: CELL CYCLE Ligands: LE9, EPE, ZN, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: LE9, EPE, ZN, PEG