Search Count: 15
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Human Tead1 In Complex With 2-(4-Chloro-3-{3-Methyl-5-[4-(Trifluoromethyl)Phenoxy]Phenyl}-1H-Pyrrolo[3,2-C]Pyridin-1-Yl)Ethan-1-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2026-02-04 Classification: TRANSCRIPTION Ligands: MYR, GOL, CL, A1JLZ |
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.50 Å Release Date: 2025-12-24 Classification: CHAPERONE Ligands: ADP |
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-11-19 Classification: CHAPERONE Ligands: ADP |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2025-04-30 Classification: ISOMERASE Ligands: A1H8Q |
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Tead1 In Complex With A Reversible Inhibitor N-[(1S)-2-Hydroxy-1-(1-Methyl-1H-Pyrazol-3-Yl)Ethyl]-2-Methyl-8-[4-(Trifluoromethyl)Phenyl]-2H,8H-Pyrazolo[3,4-B]Indole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2025-01-22 Classification: TRANSCRIPTION Ligands: GOL, A1IJL, SO4 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-04-19 Classification: ISOMERASE Ligands: IU0 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.79 Å Release Date: 2023-02-15 Classification: ISOMERASE Ligands: DMS |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2023-02-15 Classification: ISOMERASE Ligands: DMS, UPZ, 1PE |
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Human Cyclophilin D In Complex With N-(4-Aminophenyl)-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2023-02-15 Classification: ISOMERASE Ligands: V0Z, DMS |
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Human Cyclophilin D In Complex With N-(4-Aminophenyl)-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2023-02-15 Classification: ISOMERASE Ligands: UX5, DMS, PG4 |
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Human Cyclophilin D In Complex With N-[(5-Ethyl-4-Oxo-1,2,3,4,5,6- Hexahydro-1,5-Benzodiazocin-8-Yl)Methyl]-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.98 Å Release Date: 2022-09-14 Classification: ISOMERASE Ligands: DMS, 7UO |
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Optimization Of Tead P-Site Binding Fragment Hit Into In Vivo Active Lead Msc-4106
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JJU, SO4 |
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Human Tead3 In Complex With 1-Cyclopentyl-1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JIK |
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Human Cyclophilin D In Complex With N-(5-Ethyl-4-Oxo-1,2,3,4,5,6-Hexahydro-1,5-Benzodiazocin-8-Yl)-7Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2022-06-01 Classification: ISOMERASE Ligands: VDH, DMS, PG4 |
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Bone Marrow Tyrosine Kinase In Chromosome X In Complex With A Newly Designed Covalent Inhibitor Js24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-05-27 Classification: CYTOSOLIC PROTEIN Ligands: H88 |















