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Search Count: 15

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9S64 image
Human Tead1 In Complex With 2-(4-Chloro-3-{3-Methyl-5-[4-(Trifluoromethyl)Phenoxy]Phenyl}-1H-Pyrrolo[3,2-C]Pyridin-1-Yl)Ethan-1-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2026-02-04
Classification: TRANSCRIPTION
Ligands: MYR, GOL, CL, A1JLZ

9HPO image
Docedameric Ruvbl1/Ruvbl2
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Resolution:3.50 Å Release Date: 2025-12-24
Classification: CHAPERONE
Ligands: ADP

9HB4 image
Hexameric Ruvbl1/Ruvbl2 Bound To Spag1 C-Ter
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-11-19
Classification: CHAPERONE
Ligands: ADP

9F0I image
Human Cyclophilin D In Complex With Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.40 Å Release Date: 2025-04-30
Classification: ISOMERASE
Ligands: A1H8Q

9GAX image
Tead1 In Complex With A Reversible Inhibitor N-[(1S)-2-Hydroxy-1-(1-Methyl-1H-Pyrazol-3-Yl)Ethyl]-2-Methyl-8-[4-(Trifluoromethyl)Phenyl]-2H,8H-Pyrazolo[3,4-B]Indole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.93 Å Release Date: 2025-01-22
Classification: TRANSCRIPTION
Ligands: GOL, A1IJL, SO4

7ZDN image
Human Cyclophilin D In Complex With Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.55 Å Release Date: 2023-04-19
Classification: ISOMERASE
Ligands: IU0

7R2H image
0.79A Resolution Structure Of Dmso Bound Cyclophilin D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:0.79 Å Release Date: 2023-02-15
Classification: ISOMERASE
Ligands: DMS

7R2I image
Human Cyclophilin D In Complex With Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.31 Å Release Date: 2023-02-15
Classification: ISOMERASE
Ligands: DMS, UPZ, 1PE

7R2J image
Human Cyclophilin D In Complex With N-(4-Aminophenyl)-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.26 Å Release Date: 2023-02-15
Classification: ISOMERASE
Ligands: V0Z, DMS

7R2L image
Human Cyclophilin D In Complex With N-(4-Aminophenyl)-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.10 Å Release Date: 2023-02-15
Classification: ISOMERASE
Ligands: UX5, DMS, PG4

7PMT image
Human Cyclophilin D In Complex With N-[(5-Ethyl-4-Oxo-1,2,3,4,5,6- Hexahydro-1,5-Benzodiazocin-8-Yl)Methyl]-7-Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:0.98 Å Release Date: 2022-09-14
Classification: ISOMERASE
Ligands: DMS, 7UO

7ZJP image
Optimization Of Tead P-Site Binding Fragment Hit Into In Vivo Active Lead Msc-4106
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.19 Å Release Date: 2022-07-13
Classification: TRANSCRIPTION
Ligands: JJU, SO4

7ZJQ image
Human Tead3 In Complex With 1-Cyclopentyl-1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2022-07-13
Classification: TRANSCRIPTION
Ligands: JIK

7OGI image
Human Cyclophilin D In Complex With N-(5-Ethyl-4-Oxo-1,2,3,4,5,6-Hexahydro-1,5-Benzodiazocin-8-Yl)-7Methyl-2-Oxo-1H,2H-Pyrazolo[1,5-A]Pyrimidine-6-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.01 Å Release Date: 2022-06-01
Classification: ISOMERASE
Ligands: VDH, DMS, PG4

6I99 image
Bone Marrow Tyrosine Kinase In Chromosome X In Complex With A Newly Designed Covalent Inhibitor Js24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2020-05-27
Classification: CYTOSOLIC PROTEIN
Ligands: H88
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