Search Count: 20
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The Discovery Of A Novel Anticoagulant Mechanism: Factor Xi Activation Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2026-07-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1CJA, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-29
Ligands: A1CJA, NAG
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:0.99 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ACT, CA, ZN, CD, O0L |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ACT, CA, ZN, CD, O0L
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CD, O0F |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, CD, O0F
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CD, NZR |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, CD, NZR
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Ndm1-Inhibitor Co-Structure
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, NZR |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: ZN, NZR
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Ndm1-Inhibitor Co-Structure
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2023-03-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CD, ZN, NZ0, EPE |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2023-03-08
Ligands: CD, ZN, NZ0, EPE
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Hiv Reverse Transcriptase With Compound Pyr01
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2022-11-23 Classification: VIRAL PROTEIN Ligands: 9QI |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: 9QI
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Hiv Reverse Transcriptase With Compound Pyr02
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2022-11-23 Classification: VIRAL PROTEIN Ligands: 9PJ |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2022-11-23
Ligands: 9PJ
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Alpha Synuclein Fibril Formed By Full Length Protein - Rod Polymorph
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2018-09-12 Classification: PROTEIN FIBRIL |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2018-09-12
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Alpha Synuclein Fibril Formed By Full Length Protein - Twister Polymorph
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2018-09-12 Classification: PROTEIN FIBRIL |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2018-09-12
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Gpr40 In Complex With Partial Agonist Mk-8666
Organism: Homo sapiens, Enterobacteria phage t4
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-06-07 Classification: FATTY ACID BINDING PROTEIN/HYDROLASE |
Organism: Homo sapiens, Enterobacteria phage t4
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
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Gpr40 In Complex With Agopam Ap8 And Partial Agonist Mk-8666
Organism: Homo sapiens, Enterobacteria phage t4
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2017-06-07 Classification: FATTY ACID BINDING PROTEIN/HYDROLASE Ligands: OLC, MK6, 7OS |
Organism: Homo sapiens, Enterobacteria phage t4
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: OLC, MK6, 7OS
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Xfel Structure Of Human Angiotensin Ii Type 2 Receptor (Monoclinic Form) In Complex With Compound 1 (N-Benzyl-N-(2-Ethyl-4-Oxo-3-{[2'-(2H-Tetrazol-5-Yl)[1,1'-Biphenyl]-4-Yl])
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-04-05 Classification: SIGNALING PROTEIN Ligands: 8ES |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-05
Ligands: 8ES
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Xfel Structure Of Human Angiotensin Ii Type 2 Receptor (Orthorhombic Form) In Complex With Compound 1 (N-Benzyl-N-(2-Ethyl-4-Oxo-3-{[2'-(2H-Tetrazol-5-Yl)[1,1'-Biphenyl]-4-Yl] Methyl}-3,4-Dihydroquinazolin-6-Yl)Thiophene-2-Carboxamide)
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-04-05 Classification: SIGNALING PROTEIN Ligands: 8ES, OLC, OLA |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-05
Ligands: 8ES, OLC, OLA
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Synchrotron Structure Of Human Angiotensin Ii Type 2 Receptor In Complex With Compound 2 (N-[(Furan-2-Yl)Methyl]-N-(4-Oxo-2-Propyl-3-{[2'-(2H-Tetrazol-5-Yl)[1,1'- Biphenyl]-4-Yl]Methyl}-3,4-Dihydroquinazolin-6-Yl)Benzamide)
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-04-05 Classification: SIGNALING PROTEIN Ligands: 8EM |
Organism: Escherichia coli, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-05
Ligands: 8EM
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S. Aureus Mnaa-Udp Co-Structure
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2016-04-27 Classification: ISOMERASE Ligands: UDP, SO4, TRS, PG4 |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: UDP, SO4, TRS, PG4
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Selective Small Molecule Inhibition Of The Fmn Riboswitch
Organism: Fusobacterium nucleatum
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2015-10-07 Classification: RNA/INHIBITOR Ligands: K, MG, 51B |
Organism: Fusobacterium nucleatum
Method: X-RAY DIFFRACTION
Release Date: 2015-10-07
Ligands: K, MG, 51B
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Clostridium Difficile Toxin B Crop Domain In Complex With Fab Domains Of Neutralizing Antibody Bezlotoxumab
Organism: Clostridium difficile, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2014-05-21 Classification: IMMUNE SYSTEM |
Organism: Clostridium difficile, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-21
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Human Ck2 Catalytic Domain In Complex With Cx-4945
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2010-12-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3NG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-15
Ligands: 3NG, SO4
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Human Ck2 Catalytic Domain In Complex With Amppn
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2010-12-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, SO4, MG, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-15
Ligands: GOL, SO4, MG, ANP
