Search Count: 25
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Crystal Structure Of Baf60A (Smarcd1) Apo Containing Partial Coiled Coil And The Yeats-Like Domain With Topologically-Linked Swib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2026-08-05 Classification: GENE REGULATION Ligands: PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: PEG
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Co-Crystal Structure Of Baf60A (Smarcd1) In Complex With Pu.1 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2026-08-05 Classification: GENE REGULATION Ligands: EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: EDO, SO4
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Co-Crystal Structure Of Baf60A (Smarcd1) Bound To Ppsc-001
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2026-08-05 Classification: GENE REGULATION Ligands: A1CLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1CLC
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Co-Crystal Structure Of Baf60A (Smarcd1) Bound To Ppsc-002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2026-08-05 Classification: GENE REGULATION Ligands: A1CK9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1CK9
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Crystal Structure Of Pparg Ligand-Binding Domain In Complex With Ncor1 Peptide And Ftx-6746
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2026-04-22 Classification: TRANSCRIPTION Ligands: A1CCT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-22
Ligands: A1CCT
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Crystal Structure Of The P300 Acetyltransferase Domain With Allosteric Inhibitor Cpi-090 And Coa
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2019-10-23 Classification: TRANSFERASE/INHIBITOR Ligands: COA, OJ7 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: COA, OJ7
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Crystal Structure Of The P300 Acetyltransferase Domain With Allosteric Inhibitor Cpi-076 And Coa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2019-10-23 Classification: TRANSFERASE/INHIBITOR Ligands: COA, OK7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: COA, OK7
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Crystal Structure Of The Cbp Bromodomain In Complex With Cpi098
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 986, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 986, EDO
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Crystal Structure Of The Cbp Bromodomain In Complex With Cpi703
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING Ligands: 58N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 58N
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02773986
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: SCN, 68Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: SCN, 68Y
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02778174
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: EDO, SCN, 69A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: EDO, SCN, 69A
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02857790
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: ACT, CA, 69B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ACT, CA, 69B
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Cbp In Complex With Cpd23 ((R)-6-(3-(Benzyloxy)Phenyl)-4-Methyl-1,3,4,5-Tetrahydro-2H-Benzo[B][1,4]Diazepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2016-04-20 Classification: Transcription/Protein Binding Ligands: ZN, 69F, B3P, EDO, NA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ZN, 69F, B3P, EDO, NA, PEG
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Cbp In Complex With Cpd637 ((R)-4-Methyl-6-(1-Methyl-3-(1-Methyl-1H-Pyrazol-4-Yl)-1H-Indazol-5-Yl)-1,3,4,5-Tetrahydro-2H-Benzo[B][1,4]Diazepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2016-04-20 Classification: Transcription/Protein Binding Ligands: ZN, 69E, B3P, EDO, NA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ZN, 69E, B3P, EDO, NA, PEG
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Discovery Of Benzotriazolo Diazepines As Orally-Active Inhibitors Of Bet Bromodomains: Crystal Structure Of Brd4 With Cpi-13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2015-11-11 Classification: SIGNALING PROTEIN Ligands: FMT, 3X0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: FMT, 3X0
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Crystal Structure Of The First Bromodomain Of Human Brd4 Bound To Benzotriazolo-Diazepine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2015-04-08 Classification: TRANSCRIPTION Ligands: 558 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 558
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Crystal Structure Of The First Bromodomain Of Human Brd4 With Benzotriazolo-Diazepine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.06 Å Release Date: 2015-04-08 Classification: SIGNALING PROTEIN Ligands: 559 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 559
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Kutzneria Sp. 744 Ornithine N-Hydroxylase, Ktzi-Fadred-Nadp+-L-Orn
Organism: Kutzneria sp. 744
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2014-09-17 Classification: OXIDOREDUCTASE Ligands: FDA, NAP, ORN, K |
Organism: Kutzneria sp. 744
Method: X-RAY DIFFRACTION
Release Date: 2014-09-17
Ligands: FDA, NAP, ORN, K
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Kutzneria Sp. 744 Ornithine N-Hydroxylase, Ktzi-Fadox-Nadp+-L-Orn
Organism: Kutzneria sp. 744
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2014-09-17 Classification: OXIDOREDUCTASE Ligands: FAD, NAP, ORN, K |
Organism: Kutzneria sp. 744
Method: X-RAY DIFFRACTION
Release Date: 2014-09-17
Ligands: FAD, NAP, ORN, K
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Kutzneria Sp. 744 Ornithine N-Hydroxylase, Ktzi-Fadred-Ox-Nadp+-L-Orn
Organism: Kutzneria sp. 744
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2014-09-17 Classification: OXIDOREDUCTASE Ligands: FAD, NAP, ORN, K |
Organism: Kutzneria sp. 744
Method: X-RAY DIFFRACTION
Release Date: 2014-09-17
Ligands: FAD, NAP, ORN, K
