Search Count: 398
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Egfr Kinase Domain (T790Mv948R) In Complex With A Strain-Release Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2026-07-29 Classification: TRANSFERASE Ligands: EDO, A1B6E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-29
Ligands: EDO, A1B6E
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First Bromodomain Of Brdt Liganded With Inhibitor Gxh-Iv-076 (Compound 33)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2026-07-29 Classification: TRANSCRIPTION/INHIBITOR Ligands: ZNJ, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-29
Ligands: ZNJ, EDO, CL
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Brd4 Bd1 Liganded With Macrocyclic Compound 2B (Jj-Ii-352A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2025-03-19 Classification: TRANSCRIPTION Ligands: A1AAL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-19
Ligands: A1AAL, EDO
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Brd4 Bd1 Liganded With Macrocyclic Compound 2D (Jj-Ii-363A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: YPB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: YPB, EDO
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Structure Of Ddb1/Cdk12/Cyclin K With Molecular Glue Sr-4835
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.90 Å Release Date: 2024-10-16 Classification: TRANSCRIPTION Ligands: RMF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: RMF
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Crystal Structure Of Ulk1 Kinase Domain With Inhibitor Mr-2088
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2024-03-27 Classification: TRANSFERASE/INHIBITOR Ligands: WXH, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-27
Ligands: WXH, SO4, EDO
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Bromodomain Of Cbp Liganded With Inhibitor Icbp5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-02-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, YVK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-28
Ligands: EDO, YVK
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Bromodomain Of Cbp Liganded With Inhibitor Icbp2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-02-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YRI, NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-21
Ligands: YRI, NI
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Bromodomain Of Cbp Liganded With Bms-536924 And Ccs-1477
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: N6I, JHL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: N6I, JHL, EDO
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Bromodomain Of Cbp Liganded With Ccs-1477
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: PO4, JHL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: PO4, JHL, EDO
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Bromodomain Of Ep300 Liganded With Ccs-1477
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: JHL, EDO, NI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: JHL, EDO, NI, SO4
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First Bromodomain Of Brd4 Liganded With Ccs-1477
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: JHL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: JHL, EDO
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Bromodomain Of Cbp Liganded With Icbp4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: EDO, YJY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: EDO, YJY
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Bromodomain Of Cbp Liganded With Icbp6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: YID, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: YID, EDO
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Bromodomain Of Cbp Liganded With Icbp7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: YN0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: YN0, EDO
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Bromodomain Of Cbp Liganded With Icbp8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: YN5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: YN5
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Bromodomain Of Cbp Liganded With Ccs1477Int
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-01-24 Classification: TRANSFERASE Ligands: YBE, EDO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: YBE, EDO, MG
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Ternary Complex Of Cdk2 With Small Molecule Ligands Tw8672 And Dinaciclib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-05-31 Classification: Cell Cycle, Transferase Ligands: EDO, 1QK, 7TW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-31
Ligands: EDO, 1QK, 7TW
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Ternary Complex Of Cdk2 With Small Molecule Ligands Tw8672 And Roscovitine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-05-31 Classification: Cell Cycle, Transferase Ligands: EDO, RRC, 7TW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-31
Ligands: EDO, RRC, 7TW
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Cdk2 Liganded With Atp And Mg2+
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-05-31 Classification: Cell Cycle, Transferase Ligands: EDO, ATP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-31
Ligands: EDO, ATP, MG
