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4DJZ image
Catalytic Fragment Of Masp-1 In Complex With Its Specific Inhibitor Developed By Directed Evolution On Sgci Scaffold
Organism: Homo sapiens, Schistocerca gregaria
Method: X-RAY DIFFRACTION
Resolution:3.20 Å Release Date: 2012-04-25
Classification: HYDROLASE/HYDROLASE INHIBITOR

3U1J image
Aprotinin Bound To Dengue Virus Protease
Organism: Dengue virus 3, Bos taurus
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2011-11-09
Classification: HYDROLASE/HYDROLASE INHIBITOR

2R9P image
Human Mesotrypsin Complexed With Bovine Pancreatic Trypsin Inhibitor(Bpti)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Resolution:1.40 Å Release Date: 2007-12-11
Classification: hydrolase/hydrolase inhibitor
Ligands: SO4

2HI9 image
Crystal Structure Of Human Native Protein C Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2007-03-13
Classification: HYDROLASE inhibitor
Ligands: CIT, GOL

3FP6 image
Anionic Trypsin In Complex With Bovine Pancreatic Trypsin Inhibitor (Bpti) Determined To The 1.49 A Resolution Limit
Organism: Rattus norvegicus, Bos taurus
Method: X-RAY DIFFRACTION
Resolution:1.49 Å Release Date: 2009-02-17
Classification: Hydrolase/Hydrolase inhibitor
Ligands: EDO, PG4, CA, SO4

3FP8 image
Anionic Trypsin Variant S195A In Complex With Bovine Pancreatic Trypsin Inhibitor (Bpti) Determined To The 1.46 A Resolution Limit
Organism: Rattus norvegicus, Bos taurus
Method: X-RAY DIFFRACTION
Resolution:1.46 Å Release Date: 2009-02-17
Classification: Hydrolase/Hydrolase inhibitor
Ligands: EDO, PG4, CA, SO4

3FP7 image
Anionic Trypsin Variant S195A In Complex With Bovine Pancreatic Trypsin Inhibitor (Bpti) Cleaved At The Scissile Bond (Lys15-Ala16) Determined To The 1.46 A Resolution Limit
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Resolution:1.46 Å Release Date: 2009-02-17
Classification: Hydrolase/Hydrolase inhibitor
Ligands: EDO, PG4, CA, SO4

2RA3 image
Human Cationic Trypsin Complexed With Bovine Pancreatic Trypsin Inhibitor (Bpti)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Resolution:1.46 Å Release Date: 2007-12-11
Classification: hydrolase/hydrolase inhibitor
Ligands: CA, SO4

3E1Z image
Crystal Structure Of The Parasite Protesase Inhibitor Chagasin In Complex With Papain
Organism: Trypanosoma cruzi, Carica papaya
Method: X-RAY DIFFRACTION
Resolution:1.86 Å Release Date: 2009-01-27
Classification: HYDROLASE INHIBITOR/HYDROLASE
Ligands: ZN, FMT, ACY

2Z7F image
Crystal Structure Of The Complex Of Human Neutrophil Elastase With 1/2Slpi
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2008-08-26
Classification: Hydrolase/Hydrolase inhibitor

2CIO image
The High Resolution X-Ray Structure Of Papain Complexed With Fragments Of The Trypanosoma Brucei Cysteine Protease Inhibitor Icp.
Organism: Trypanosoma brucei, Carica papaya
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2006-05-18
Classification: HYDROLASE/INHIBITOR
Ligands: GOL, ACT

5TG2 image
1.75 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The A N-Pentyl Substituted Macrocyclic Inhibitor (17-Mer)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Resolution:1.75 Å Release Date: 2017-01-11
Classification: PROTEASE/PROTEASE INHIBITOR
Ligands: V69

5TG1 image
1.40 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The A M-Chlorophenyl Substituted Macrocyclic Inhibitor (17-Mer)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Resolution:1.40 Å Release Date: 2017-01-11
Classification: PROTEASE/PROTEASE INHIBITOR
Ligands: CL, V56

3GYM image
Structure Of Prostasin In Complex With Aprotinin
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2009-05-05
Classification: HYDROLASE/INHIBITOR

4ISO image
Crystal Structure Of Matriptase In Complex With Its Inhibitor Hai-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.01 Å Release Date: 2013-03-06
Classification: hydrolase/hydrolase inhibitor
Ligands: GSH, GOL, PEG, PGE

4ISL image
Crystal Structure Of The Inactive Matriptase In Complex With Its Inhibitor Hai-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.29 Å Release Date: 2013-03-06
Classification: hydrolase/hydrolase inhibitor
Ligands: PG4, GOL, PGE, GSH

5E0J image
1.20 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (21-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Resolution:1.20 Å Release Date: 2016-05-04
Classification: PROTEASE/PROTEASE INHIBITOR
Ligands: CL, 5LJ

5E0H image
1.95 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (18-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2016-05-04
Classification: PROTEASE/PROTEASE INHIBITOR
Ligands: 5LH, GOL

5E0G image
1.20 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (17-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION
Resolution:1.20 Å Release Date: 2016-05-04
Classification: PROTEASE/PROTEASE INHIBITOR
Ligands: CL, 5LG

1QLQ image
Bovine Pancreatic Trypsin Inhibitor (Bpti) Mutant With Altered Binding Loop Sequence
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Resolution:1.42 Å Release Date: 1999-10-05
Classification: SERINE PROTEASE INHIBITOR
Ligands: SO4
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