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Catalytic Fragment Of Masp-1 In Complex With Its Specific Inhibitor Developed By Directed Evolution On Sgci Scaffold
Organism: Homo sapiens, Schistocerca gregaria
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2012-04-25 Classification: HYDROLASE/HYDROLASE INHIBITOR |
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Organism: Dengue virus 3, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR |
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Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2007-12-11 Classification: hydrolase/hydrolase inhibitor Ligands: SO4 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-03-13 Classification: HYDROLASE inhibitor Ligands: CIT, GOL |
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Anionic Trypsin In Complex With Bovine Pancreatic Trypsin Inhibitor (Bpti) Determined To The 1.49 A Resolution Limit
Organism: Rattus norvegicus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2009-02-17 Classification: Hydrolase/Hydrolase inhibitor Ligands: EDO, PG4, CA, SO4 |
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Anionic Trypsin Variant S195A In Complex With Bovine Pancreatic Trypsin Inhibitor (Bpti) Determined To The 1.46 A Resolution Limit
Organism: Rattus norvegicus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2009-02-17 Classification: Hydrolase/Hydrolase inhibitor Ligands: EDO, PG4, CA, SO4 |
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Anionic Trypsin Variant S195A In Complex With Bovine Pancreatic Trypsin Inhibitor (Bpti) Cleaved At The Scissile Bond (Lys15-Ala16) Determined To The 1.46 A Resolution Limit
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2009-02-17 Classification: Hydrolase/Hydrolase inhibitor Ligands: EDO, PG4, CA, SO4 |
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Human Cationic Trypsin Complexed With Bovine Pancreatic Trypsin Inhibitor (Bpti)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2007-12-11 Classification: hydrolase/hydrolase inhibitor Ligands: CA, SO4 |
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Crystal Structure Of The Parasite Protesase Inhibitor Chagasin In Complex With Papain
Organism: Trypanosoma cruzi, Carica papaya
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2009-01-27 Classification: HYDROLASE INHIBITOR/HYDROLASE Ligands: ZN, FMT, ACY |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2008-08-26 Classification: Hydrolase/Hydrolase inhibitor |
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The High Resolution X-Ray Structure Of Papain Complexed With Fragments Of The Trypanosoma Brucei Cysteine Protease Inhibitor Icp.
Organism: Trypanosoma brucei, Carica papaya
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2006-05-18 Classification: HYDROLASE/INHIBITOR Ligands: GOL, ACT |
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1.75 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The A N-Pentyl Substituted Macrocyclic Inhibitor (17-Mer)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2017-01-11 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: V69 |
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1.40 A Resolution Structure Of Norovirus 3Cl Protease In Complex With The A M-Chlorophenyl Substituted Macrocyclic Inhibitor (17-Mer)
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-01-11 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: CL, V56 |
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Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-05-05 Classification: HYDROLASE/INHIBITOR |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: GSH, GOL, PEG, PGE |
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Crystal Structure Of The Inactive Matriptase In Complex With Its Inhibitor Hai-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: PG4, GOL, PGE, GSH |
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1.20 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (21-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2016-05-04 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: CL, 5LJ |
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1.95 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (18-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-05-04 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: 5LH, GOL |
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1.20 A Resolution Structure Of Norovirus 3Cl Protease In Complex With A Triazole-Based Macrocyclic (17-Mer) Inhibitor
Organism: Norwalk virus
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2016-05-04 Classification: PROTEASE/PROTEASE INHIBITOR Ligands: CL, 5LG |
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Bovine Pancreatic Trypsin Inhibitor (Bpti) Mutant With Altered Binding Loop Sequence
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 1999-10-05 Classification: SERINE PROTEASE INHIBITOR Ligands: SO4 |




















