Search Count: 20
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Structure Of Plasmodium Falciparum 20S Proteasome Bound To An Asparagine-Ethylenediamine Based Inhibitor Tdi6245
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY Resolution:2.86 Å Release Date: 2026-07-29 Classification: HYDROLASE Ligands: A1CRS |
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY
Release Date: 2026-07-29
Ligands: A1CRS
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Crystal Structure Of An Inverse Agonist Antipsychotic Drug Derivative-Bound 5-Ht2C
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2024-08-28 Classification: MEMBRANE PROTEIN Ligands: A1L10 |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2024-08-28
Ligands: A1L10
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Crystal Structure Of An Inverse Agonist Antipsychotic Drug Pimavanserin-Bound 5-Ht2A
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2024-08-28 Classification: MEMBRANE PROTEIN Ligands: A1L11 |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2024-08-28
Ligands: A1L11
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Macrocyclic Peptides Tdi5575 That Selectively Inhibit The Mycobacterium Tuberculosis Proteasome
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-04-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: U5Y, CIT, DMF |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2021-04-28
Ligands: U5Y, CIT, DMF
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Structure Of Mtb Lpd Bound To 010705
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2021-01-27 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: FAD, WPM, GOL |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2021-01-27
Ligands: FAD, WPM, GOL
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P38 In Complex With T-3220137
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-11-20 Classification: TRANSFERASE/INHIBITOR Ligands: MKP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: MKP
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor A85
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMF, M6M, CIT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: DMF, M6M, CIT
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor A86
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMF, M6Y, CIT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: DMF, M6Y, CIT
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor B6
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: M9G |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: M9G
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Integrin Alphavbeta3 Ectodomain Bound To Antagonist Tdi-4161
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2019-09-25 Classification: CELL ADHESION Ligands: NAG, MN, JUY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: NAG, MN, JUY
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Human Cgas Catalytic Domain Bound With The Inhibitor G108
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: JUM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-29
Ligands: JUM, ZN
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Human Cgas Catalytic Domain Bound With The Inhibitor G150
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2019-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, JUJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-29
Ligands: ZN, JUJ
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Human Cgas Catalytic Domain Bound With Cgamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1SY, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-29
Ligands: 1SY, ZN
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[4,5-B]Pyridine-2-One Based P38 Map Kinase Inhibitors By Scaffold Hopping: Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-04-17 Classification: TRANSFERASE Ligands: J8S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: J8S
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[4,5-B]Pyridine-2-One Based P38 Map Kinase Inhibitors By Scaffold Hopping - Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-04-17 Classification: TRANSFERASE/INHIBITOR Ligands: J9G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: J9G
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Mouse Cgas Bound To The Inhibitor Ru332
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2017-10-11 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: ZN, AE7 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-10-11
Ligands: ZN, AE7
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Mouse Cgas Bound To The Inhibitor Ru521
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2017-10-11 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: ZN, AEV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-10-11
Ligands: ZN, AEV
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Mouse Cgas Bound To The Inhibitor Ru365
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2017-08-09 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: ZN, A9Y |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: ZN, A9Y
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X-Ray Crystal Structure Of Racemic Non-Glycosylated Chemokine Ser-Ccl1
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-05-07 Classification: SIGNALING PROTEIN Ligands: SO4 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: SO4
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(Quasi-)Racemic X-Ray Crystal Structure Of Glycosylated Chemokine Ser-Ccl1.
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-05-07 Classification: SIGNALING PROTEIN Ligands: NAG, SO4, CIT |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: NAG, SO4, CIT