Search Count: 70
![]() |
Probing 3-Amino-2H-Azaindazoles As Allosteric Inhibitors Of The Protein Tyrosine Phosphatase Shp2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2026-06-24 Classification: PEPTIDE BINDING PROTEIN Ligands: A1JWM, ACT, EDO, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-24
Ligands: A1JWM, ACT, EDO, NA
![]() |
Mapping The Shp2 Allosteric Pocket With Target-Biased Covalent Fragments
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2026-05-06 Classification: CYTOSOLIC PROTEIN Ligands: EDO, A1JWN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-06
Ligands: EDO, A1JWN
![]() |
Langerin In Complex With Thiazolopyrimidine
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2026-02-25 Classification: SUGAR BINDING PROTEIN Ligands: A1JHV, CA |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2026-02-25
Ligands: A1JHV, CA
![]() |
Structure Of The Mus Musclus Langerin Carbohydrate Recognition Domain With Depleted Calcium
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2025-11-19 Classification: IMMUNE SYSTEM Ligands: CL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2025-11-19
Ligands: CL
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 2 In Complex With Inhibitor Ag-01-128
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2025-07-16 Classification: METAL BINDING PROTEIN Ligands: FE, JCR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-16
Ligands: FE, JCR
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 2 In Complex With Inhibitor Km-06-098
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2025-07-16 Classification: METAL BINDING PROTEIN Ligands: FE, UVU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-16
Ligands: FE, UVU
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 1 In Complex With Inhibitor Lp778902
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2025-07-16 Classification: METAL BINDING PROTEIN Ligands: FE, A1IT9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-16
Ligands: FE, A1IT9
![]() |
Crystal Structure Of Monoacylglycerol Lipase With Bodipy Labeled Probe
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2025-06-11 Classification: HYDROLASE Ligands: A1IIH, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: A1IIH, EDO
![]() |
Crystal Structure Of Human Monoglyceride Lipase In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2025-02-12 Classification: HYDROLASE Ligands: A1H35, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1H35, EDO
![]() |
Crystal Structure Of Human Monoacylglycerol Lipase With Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2024-12-11 Classification: HYDROLASE Ligands: A1IG3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-11
Ligands: A1IG3, EDO
![]() |
Clathrin Terminal Domain Complexed With Pitstop 2C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2024-06-26 Classification: ENDOCYTOSIS Ligands: DMS, PEG, EDO, GOL, ACT, A1ATR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: DMS, PEG, EDO, GOL, ACT, A1ATR
![]() |
Clathrin Terminal Domain Complexed With Pitstop 2D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2024-06-26 Classification: ENDOCYTOSIS Ligands: DMS, TRS, PEG, ACT, EDO, GOL, A1ATQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: DMS, TRS, PEG, ACT, EDO, GOL, A1ATQ
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 1 In Complex With Inhibitor Km-07-052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2024-01-10 Classification: METAL BINDING PROTEIN Ligands: FE, UWC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: FE, UWC
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 1 In Complex With Inhibitor Km-06-057
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2024-01-10 Classification: METAL BINDING PROTEIN Ligands: FE, UVF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: FE, UVF
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 1 In Complex With Inhibitor Km-06-098
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2024-01-10 Classification: METAL BINDING PROTEIN Ligands: FE, UVU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: FE, UVU
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 1 In Complex With Inhibitor Tpt-004
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2024-01-10 Classification: METAL BINDING PROTEIN Ligands: FE, UXC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: FE, UXC
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 1 In Complex With Inhibitor Km-07-047
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-01-10 Classification: METAL BINDING PROTEIN Ligands: FE, UXL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: FE, UXL
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 1 In Complex With Inhibitor Km-06-070
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2024-01-10 Classification: METAL BINDING PROTEIN Ligands: FE, UX3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: FE, UX3
![]() |
Crystal Structure Of Human Tryptophan Hydroxylase 1 In Complex With Inhibitor Km-06-004
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2024-01-10 Classification: METAL BINDING PROTEIN Ligands: FE, UWL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: FE, UWL
![]() |
Tankyrase 2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-10-11 Classification: TRANSFERASE Ligands: OY6, SO4, ZN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: OY6, SO4, ZN, GOL
