Search Count: 41
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Crystal Structure Of Selective Inhibitor 16 Bound At The Active Site Of Cdk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-07-08 Classification: SIGNALING PROTEIN Ligands: A1DEQ, A1DJL, GOL, SO4, DMS, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: A1DEQ, A1DJL, GOL, SO4, DMS, EPE
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Structure Of Cbl-B Bound To Compound 33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-07-01 Classification: LIGASE Ligands: GOL, IOD, EDO, MG, ZN, A1DCD, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: GOL, IOD, EDO, MG, ZN, A1DCD, DMS
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Structure Of C-Cbl Bound To Compound 33
Organism: Schistosoma japonicum, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2026-07-01 Classification: LIGASE Ligands: A1DCD, ZN, MG |
Organism: Schistosoma japonicum, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: A1DCD, ZN, MG
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Plk4 In Complex With Compound 6 (3-Hydroxy-N-(3-(Pyridin-2-Yl)-1H-Pyrazol-4-Yl)-8-Azabicyclo[3.2.1]Octane-8-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2026-02-18 Classification: TRANSFERASE Ligands: SO4, A1CTX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: SO4, A1CTX
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Plk4 In Complex With Compound 25 ((R)-7-Hydroxy-N-(3-(1-(2,2,2-Trifluoroethyl)-1H-Pyrazolo[4,3-C]Pyridin-6-Yl)-1H-Pyrazol-4-Yl)-7-(Trifluoromethyl)-4-Azaspiro[2.5]Octane-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2026-02-18 Classification: TRANSFERASE Ligands: A1CTV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: A1CTV, SO4
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Cyclin-Free Cdk2 In Complex With Cpd17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2023-10-18 Classification: TRANSFERASE Ligands: WQ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-18
Ligands: WQ6
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Cyclin-Free Cdk2 In Complex With Cpd21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2023-10-18 Classification: TRANSFERASE Ligands: GOL, WQK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-18
Ligands: GOL, WQK
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Ccbl Tkb Domain In Complex With Pzap70 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2022-11-09 Classification: IMMUNE SYSTEM Ligands: MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: MG
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Cryoem Structure Of The Smc5/6-Holocomplex (Composite Structure)
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: ELECTRON MICROSCOPY Release Date: 2022-09-21 Classification: RECOMBINATION Ligands: ZN |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: ELECTRON MICROSCOPY
Release Date: 2022-09-21
Ligands: ZN
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Ternary Complex Of Vhl/Brd4-Bd1/Compound9 (4-(3,5-Difluoropyridin-2-Yl)-N-(11-(((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-Methylthiazol-5-Yl)Benzyl)Carbamoyl)Pyrrolidin-1-Yl)-3,3-Dimethyl-1-Oxobutan-2-Yl)Amino)-11-Oxoundecyl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-02-24 Classification: PEPTIDE BINDING PROTEIN Ligands: WEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: WEP
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Brd4-Bd1 Compound6 (Methyl 4-(3,5-Difluoropyridin-2-Yl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2021-02-24 Classification: CELL CYCLE Ligands: WEM, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: WEM, GOL
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Pim1 In Complex With Cpd9 ((R)-5-Amino-N-(3-(4-Aminoazepan-1-Yl)-1H-Pyrazol-4-Yl)-2-(2,6-Difluorophenyl)Thiazole-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2019-11-27 Classification: TRANSFERASE Ligands: KUY, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: KUY, PO4
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Crebbp Bromodomain In Complex With Cpd 30 (1-(3-(3-(1-Methyl-1H-Pyrazol-4-Yl)Isoquinolin-8-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-10-17 Classification: PROTEIN BINDING/INHIBITOR Ligands: ZN, B3P, BKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: ZN, B3P, BKJ
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Brd4-Bd1 In Complex With Cpd19 (3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridine-5-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2018-05-30 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: EDO, 9U4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: EDO, 9U4
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Usp7 In Complex With Cpd2 (4-(3-(1-Methylpiperidin-4-Yl)-1,2,4-Oxadiazol-5-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2017-12-13 Classification: HYDROLASE Ligands: AJJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: AJJ, GOL
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Pi3K-Gamma K802T In Complex With Cpd 8 10-((1-(Tert-Butyl)Piperidin-4-Yl)Sulfinyl)-2-(1-Isopropyl-1H-1,2,4-Triazol-5-Yl)-5,6-Dihydrobenzo[F]Imidazo[1,2-D][1,4]Oxazepine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2017-11-15 Classification: TRANSFERASE/TRANSFERASE INHBITOR Ligands: BWY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: BWY
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Crystal Structure Of The C-Terminal Domain Of Doublecortin (Tgdcx) From Toxoplasma Gondii Me49
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-10-18 Classification: STRUCTURAL PROTEIN Ligands: FMT |
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: FMT
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Structural Insights Into Lipoprotein N-Acylation By Escherichia Coli Apolipoprotein N-Acyltransferase
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2017-07-12 Classification: TRANSFERASE Ligands: OLC, LNK, PLM, CL |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: OLC, LNK, PLM, CL
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Apolipoprotein N-Acyltransferase C387S Active Site Mutant
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2017-07-12 Classification: TRANSFERASE Ligands: OLB, MG, PLM, CL, OLC |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: OLB, MG, PLM, CL, OLC
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Crystal Structure Of The S.Pombe Smc5/6 Hinge Domain
Organism: Schizosaccharomyces pombe
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-02-08 Classification: RECOMBINATION Ligands: SO4, GOL |
Organism: Schizosaccharomyces pombe
Method: X-RAY DIFFRACTION
Release Date: 2017-02-08
Ligands: SO4, GOL
