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11GV image
Crystal Structure Of Selective Inhibitor 16 Bound At The Active Site Of Cdk2

11GY image
Crystal Structure Of Selective Inhibitor 16 Bound At The Active Site Of Cdk1

10YS image
Structure Of Cbl-B Bound To Compound 33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2026-07-01
Classification: LIGASE
Ligands: GOL, IOD, EDO, MG, ZN, A1DCD, DMS

10ZF image
Structure Of C-Cbl Bound To Compound 33

9Y9B image
Plk4 In Complex With Compound 6 (3-Hydroxy-N-(3-(Pyridin-2-Yl)-1H-Pyrazol-4-Yl)-8-Azabicyclo[3.2.1]Octane-8-Carboxamide)

9Y9N image
Plk4 In Complex With Compound 25 ((R)-7-Hydroxy-N-(3-(1-(2,2,2-Trifluoroethyl)-1H-Pyrazolo[4,3-C]Pyridin-6-Yl)-1H-Pyrazol-4-Yl)-7-(Trifluoromethyl)-4-Azaspiro[2.5]Octane-4-Carboxamide)

8ERD image
Cyclin-Free Cdk2 In Complex With Cpd17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.33 Å Release Date: 2023-10-18
Classification: TRANSFERASE
Ligands: WQ6

8ERN image
Cyclin-Free Cdk2 In Complex With Cpd21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.64 Å Release Date: 2023-10-18
Classification: TRANSFERASE
Ligands: GOL, WQK

7SIY image
Ccbl Tkb Domain In Complex With Pzap70 Peptide

7QCD image
Cryoem Structure Of The Smc5/6-Holocomplex (Composite Structure)

7KHH image
Ternary Complex Of Vhl/Brd4-Bd1/Compound9 (4-(3,5-Difluoropyridin-2-Yl)-N-(11-(((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-Methylthiazol-5-Yl)Benzyl)Carbamoyl)Pyrrolidin-1-Yl)-3,3-Dimethyl-1-Oxobutan-2-Yl)Amino)-11-Oxoundecyl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxamide)

7KHL image
Brd4-Bd1 Compound6 (Methyl 4-(3,5-Difluoropyridin-2-Yl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.29 Å Release Date: 2021-02-24
Classification: CELL CYCLE
Ligands: WEM, GOL

6NO8 image
Pim1 In Complex With Cpd9 ((R)-5-Amino-N-(3-(4-Aminoazepan-1-Yl)-1H-Pyrazol-4-Yl)-2-(2,6-Difluorophenyl)Thiazole-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.38 Å Release Date: 2019-11-27
Classification: TRANSFERASE
Ligands: KUY, PO4

6ALB image
Crebbp Bromodomain In Complex With Cpd 30 (1-(3-(3-(1-Methyl-1H-Pyrazol-4-Yl)Isoquinolin-8-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5VZS image
Brd4-Bd1 In Complex With Cpd19 (3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridine-5-Carboxamide)

5WHC image
Usp7 In Complex With Cpd2 (4-(3-(1-Methylpiperidin-4-Yl)-1,2,4-Oxadiazol-5-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2017-12-13
Classification: HYDROLASE
Ligands: AJJ, GOL

6AUD image
Pi3K-Gamma K802T In Complex With Cpd 8 10-((1-(Tert-Butyl)Piperidin-4-Yl)Sulfinyl)-2-(1-Isopropyl-1H-1,2,4-Triazol-5-Yl)-5,6-Dihydrobenzo[F]Imidazo[1,2-D][1,4]Oxazepine

6B4A image
Crystal Structure Of The C-Terminal Domain Of Doublecortin (Tgdcx) From Toxoplasma Gondii Me49

5VRG image
Structural Insights Into Lipoprotein N-Acylation By Escherichia Coli Apolipoprotein N-Acyltransferase

5VRH image
Apolipoprotein N-Acyltransferase C387S Active Site Mutant
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