Search Count: 15
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Structure Of Plasmodium Falciparum 20S Proteasome Bound To An Asparagine-Ethylenediamine Based Inhibitor Tdi6245
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY Resolution:2.86 Å Release Date: 2026-07-29 Classification: HYDROLASE Ligands: A1CRS |
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY
Release Date: 2026-07-29
Ligands: A1CRS
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Nsp14 In Complex With Ligand Tdi-016037-Nx-1
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2025-08-27 Classification: VIRAL PROTEIN Ligands: ZN, SAH, A1JDF, CL, EDO, IMD, IPA, SO4 |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2025-08-27
Ligands: ZN, SAH, A1JDF, CL, EDO, IMD, IPA, SO4
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Co-Crystal Structure Of Optimized Analog Tdi-13537 Provided New Insights Into The Potency Determinants Of The Sulfonamide Inhibitor Series
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2024-01-03 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: FAD, U4I, GOL |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2024-01-03
Ligands: FAD, U4I, GOL
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Cryo-Em Structure Of Mtb Lpd Bound To Inhibitor Complex With 2-((2-Cyano-N,5-Dimethyl-1H-Indole)-7-Sulfonamido)-N-(4-(Oxetan-3-Yl)-3,4-Dihydro-2H-Benzo[B] [1,4]Oxazin-7-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: ELECTRON MICROSCOPY Release Date: 2022-05-25 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: FAD, OU6 |
Organism: Mycobacterium tuberculosis
Method: ELECTRON MICROSCOPY
Release Date: 2022-05-25
Ligands: FAD, OU6
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Human Soluble Adenylyl Cyclase In Complex With The Inhibitor Tdi10229
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-10-06 Classification: SIGNALING PROTEIN Ligands: 1S2, ACT, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 1S2, ACT, DMS, EDO
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Macrocyclic Peptides Tdi5575 That Selectively Inhibit The Mycobacterium Tuberculosis Proteasome
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-04-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: U5Y, CIT, DMF |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2021-04-28
Ligands: U5Y, CIT, DMF
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Structure Of Mtb Lpd Bound To 010705
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2021-01-27 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: FAD, WPM, GOL |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2021-01-27
Ligands: FAD, WPM, GOL
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor A85
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMF, M6M, CIT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: DMF, M6M, CIT
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor A86
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMF, M6Y, CIT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: DMF, M6Y, CIT
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Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor B6
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: M9G |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: M9G
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Crystal Structure Of Human Phgdh Complexed With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-07-24 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: ONV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: ONV, EDO
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Crystal Structure Of Human Phgdh Complexed With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2019-07-24 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: ONS, MLT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: ONS, MLT
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Human Cgas Catalytic Domain Bound With The Inhibitor G108
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: JUM, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-29
Ligands: JUM, ZN
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Human Cgas Catalytic Domain Bound With The Inhibitor G150
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2019-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, JUJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-29
Ligands: ZN, JUJ
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Human Cgas Catalytic Domain Bound With Cgamp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1SY, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-29
Ligands: 1SY, ZN