Search Count: 20
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Cryoem Structure Of Mu-Opioid Receptor - Gi Protein Complex Bound To Fluornitrazene (Fnz)
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY Release Date: 2026-04-01 Classification: MEMBRANE PROTEIN Ligands: A1B79 |
Organism: Homo sapiens, Mus musculus
Method: ELECTRON MICROSCOPY
Release Date: 2026-04-01
Ligands: A1B79
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Outward-Open Structure Of Human Glycine Transporter 2 Bound To Allosteric Inhibitor Org25543
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:2.49 Å Release Date: 2026-02-25 Classification: MEMBRANE PROTEIN Ligands: A1EF1, Y01, CLR, CL, NA |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-02-25
Ligands: A1EF1, Y01, CLR, CL, NA
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Outward-Open Structure Of Human Glycine Transporter 2 Bound To Allosteric Inhibitor Rpi-Glyt2-82
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-02-25 Classification: MEMBRANE PROTEIN Ligands: CL, A1IXX, CLR, Y01, NA |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-02-25
Ligands: CL, A1IXX, CLR, Y01, NA
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Inward-Open Structure Of Human Glycine Transporter 2 In Substrate-Free State
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-02-25 Classification: MEMBRANE PROTEIN Ligands: CLR, CL |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-02-25
Ligands: CLR, CL
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Inward-Occluded Structure Of Human Glycine Transporter 2 Bound To Substrate Glycine
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2026-02-25 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-02-25
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Crystal Structure Of The Mertk Kinase Domain With Sa4488
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-10-09 Classification: TRANSFERASE Ligands: A1APF, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APF, CL
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Mertk In Complex With Small Molecule 6-{1-[([1,1'-Biphenyl]-4-Yl)Carbamoyl]Azetidin-3-Yl}-3-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2024-10-09 Classification: TRANSFERASE/INHIBITOR Ligands: A1APG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APG, CL
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Mertk In Complex With Small Molecule Inhibitor 6-{1-[6-(3-Hydroxy-3-Methylbutoxy)-1,3-Benzoxazol-2-Yl]Azetidin-3-Yl}-3-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2024-10-09 Classification: TRANSFERASE/INHIBITOR Ligands: A1APH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APH, CL
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Discovery Of Spirohydantoins As Selective, Orally Bioavailable Inhibitors Of P300/Cbp Histone Acetyltransferases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2021-03-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Y2P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-17
Ligands: Y2P
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The Novel P300/Cbp Inhibitor A-485 Uncovers A Unique Mechanism Of Action To Target Ar In Castrate Resistant Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-09-27 Classification: transferase/transferase INHIBITOR Ligands: 6TF, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: 6TF, NA
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Crystal Structure Of Human Nampt With A-1293201
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: 7T7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7T7, SO4
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Crystal Structure Of Human Nampt With A-1326133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 7TA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: SO4, 7TA
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HY
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HV
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Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(2-Methoxyphenyl)Methyl]-N,N-Dimethyl-4-(1-Methylindol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING, INHIBITOR Ligands: LQD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: LQD
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Polycomb Protein Eed In Complex With Inhibitor: 2-[4-(4-{(3S,4R)-4-(Dimethylamino)-1-[(2-Fluoro-6-Methylphenyl)Methyl]Pyrrolidin-3-Yl}Phenyl)-1H-Pyrazol-1-Yl]Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING, INHIBITOR Ligands: 7XG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 7XG
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Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(2-Bromo-6-Fluorophenyl)Methyl]-N,N-Dimethyl-4-(1-Methyl-1H-Indol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: 82D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 82D
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Polycomb Protein Eed In Complex With Inhibitor: (3R,4S)-1-[(1S)-7-Fluoro-2,3-Dihydro-1H-Inden-1-Yl]-N,N-Dimethyl-4-(1-Methyl-1H-Indol-3-Yl)Pyrrolidin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2017-03-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: 82G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 82G
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The Novel Suv4-20 Inhibitor A-196 Verifies A Role For Epigenetics In Genomic Integrity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2017-01-25 Classification: TRANSFERASE Ligands: ZN, SAM, 539 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: ZN, SAM, 539
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Human G9A In Complex With Inhibitor A-366
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2014-01-15 Classification: Transferase/Transferase Inhibitor Ligands: 2OD, SAH, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-15
Ligands: 2OD, SAH, ZN