Search Count: 26
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Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Compound 7, A Novel Nanomolar A2A Receptor Antagonist From Modern Hit-Finding With Structure-Guided De Novo Design
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2025-06-18 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
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Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Compound 9, A Novel Nanomolar A2A Receptor Antagonist From Modern Hit-Finding With Structure-Guided De Novo Design
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2025-06-18 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
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Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Chromone 4D
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2020-09-16 Classification: PROTEIN BINDING Ligands: QGE, NA, CLR, OLA, OLC |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: QGE, NA, CLR, OLA, OLC
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Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Chromone 5D
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2020-09-16 Classification: PROTEIN BINDING Ligands: QGW, NA, CLR, OLB, OLA, OLC |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: QGW, NA, CLR, OLB, OLA, OLC
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Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer With Bound High Affinity Inhibitor
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-07-15 Classification: MEMBRANE PROTEIN Ligands: QLQ, PG4 |
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-15
Ligands: QLQ, PG4
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Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer With Bound High Affinity Inhibitor
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2020-07-15 Classification: MEMBRANE PROTEIN Ligands: PG4, 3N6 |
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-15
Ligands: PG4, 3N6
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Crystal Structure Of The Orexin-1 Receptor In Complex With Gsk1059865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2020-01-15 Classification: MEMBRANE PROTEIN Ligands: NRE, PG4, CIT, SO4, SOG, NA, PGW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: NRE, PG4, CIT, SO4, SOG, NA, PGW
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Crystal Structure Of The Orexin-1 Receptor In Complex With Lemborexant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2020-01-15 Classification: MEMBRANE PROTEIN Ligands: NRK, PG4, SO4, SOG, PGW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: NRK, PG4, SO4, SOG, PGW
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Crystal Structure Of The Orexin-1 Receptor In Complex With Suvorexant At 2.29 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: SUV, PG4, CIT, SOG, PGW, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: SUV, PG4, CIT, SOG, PGW, NA
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Crystal Structure Of The Orexin-1 Receptor In Complex With Empa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: 7MA, SO4, PG4, CIT, SOG, PGW, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: 7MA, SO4, PG4, CIT, SOG, PGW, NA
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Crystal Structure Of The Orexin-1 Receptor In Complex With Daridorexant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: NS2, SO4, PGW, SOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NS2, SO4, PGW, SOG
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Crystal Structure Of The Orexin-1 Receptor In Complex With Act-462206
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: NRZ, SOG, SO4, PGW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NRZ, SOG, SO4, PGW
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Crystal Structure Of The Orexin-1 Receptor In Complex With Filorexant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: NT5, PG4, SO4, SOG, CL, PGW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NT5, PG4, SO4, SOG, CL, PGW
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Crystal Structure Of The Orexin-2 Receptor In Complex With Empa At 2.74 A Resolution
Organism: Homo sapiens, Pyrococcus abyssi ge5
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: 7MA, PG4, OLA |
Organism: Homo sapiens, Pyrococcus abyssi ge5
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: 7MA, PG4, OLA
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Crystal Structure Of The Orexin-2 Receptor In Complex With Suvorexant At 2.76 A Resolution
Organism: Homo sapiens, Pyrococcus abyssi ge5
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: OLA, SUV, NH4, PG4 |
Organism: Homo sapiens, Pyrococcus abyssi ge5
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: OLA, SUV, NH4, PG4
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Crystal Structure Of The Orexin-2 Receptor In Complex With Htl6641 At 2.61 A Resolution
Organism: Homo sapiens, Pyrococcus abyssi (strain ge5 / orsay)
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: NU8, NO3, PG4, OLA |
Organism: Homo sapiens, Pyrococcus abyssi (strain ge5 / orsay)
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NU8, NO3, PG4, OLA
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Crystal Structure Of The Orexin-1 Receptor In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: NV8, SO4, PGW, SOG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NV8, SO4, PGW, SOG, NA
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Crystal Structure Of The Orexin-1 Receptor In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: NVH, SO4, PGW, SOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NVH, SO4, PGW, SOG, PG4
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Crystal Structure Of The Orexin-1 Receptor In Complex With Sb-334867
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: NVK, SO4, SOG, PGW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NVK, SO4, SOG, PGW
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Crystal Structure Of The Orexin-1 Receptor In Complex With Sb-408124
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2020-01-01 Classification: MEMBRANE PROTEIN Ligands: NVN, SOG, SO4, PGW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: NVN, SOG, SO4, PGW
