Search Count: 13
![]() |
Structure Of Gpr61 Bound To Inverse Agonist Compound 15
Organism: Homo sapiens, Lama glama
Method: ELECTRON MICROSCOPY Resolution:3.08 Å Release Date: 2026-03-25 Classification: SIGNALING PROTEIN Ligands: A1CWB |
Organism: Homo sapiens, Lama glama
Method: ELECTRON MICROSCOPY
Release Date: 2026-03-25
Ligands: A1CWB
![]() |
Design And Application Of Synthetic 17B-Hsd13 Substrates To Drug Discovery, And To Reveal Preserved Catalytic Activity Of Protective Human Variants
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2024-11-27 Classification: HYDROLASE Ligands: NAD, A1AG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: NAD, A1AG4
![]() |
Design And Application Of Synthetic 17B-Hsd13 Substrates To Drug Discovery, And To Reveal Preserved Catalytic Activity Of Protective Human Variants
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2024-11-27 Classification: HYDROLASE Ligands: NAD, A1AG5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: NAD, A1AG5
![]() |
Design And Application Of Synthetic 17B-Hsd13 Substrates To Drug Discovery, And To Reveal Preserved Catalytic Activity Of Protective Human Variants
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2024-11-27 Classification: HYDROLASE Ligands: NAD, A1AG6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: NAD, A1AG6
![]() |
Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A4G, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A4G, SO4
![]() |
Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A1Y, SO4, CIT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A1Y, SO4, CIT, GOL
![]() |
Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A2J, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A2J, SO4, GOL
![]() |
Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A3J, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A3J, SO4, CL
![]() |
Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A3Y, SO4, CIT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A3Y, SO4, CIT, GOL
![]() |
Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A4J, SO4, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A4J, SO4, CIT
![]() |
Human Cytochrome P450 2D6 Bace1 Inhibitor 5 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-05-20 Classification: OXIDOREDUCTASE Ligands: HEM, SI5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-20
Ligands: HEM, SI5, ZN
![]() |
Human Cytochrome P450 2D6 Bace1 Inhibitor 6 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-05-20 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: HEM, SI6, ZN, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-20
Ligands: HEM, SI6, ZN, GOL, NA
![]() |
Crystal Structure Of Bace1 With A Pyrazole-Substituted Tetrahydropyran Thioamidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-04-01 Classification: hydrolase/hydrolase inhibitor Ligands: SI5, IOD, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-01
Ligands: SI5, IOD, GOL, DMS
