Search Count: 36
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Type-Iii C-Met Inhibitor Enabled By Free-Energy Perturbation Calculations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2026-05-27 Classification: TRANSFERASE Ligands: A1C9B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1C9B
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Engineered Ascas12A (M537R, F870L)
Organism: Acidaminococcus
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2025-12-24 Classification: SPLICING/DNA/RNA |
Organism: Acidaminococcus
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
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Abl Kinase In Complex With Ski And Asciminib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2023-09-06 Classification: TRANSFERASE Ligands: AY7, SKI, CL, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: AY7, SKI, CL, SO4, DMS
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Aura Bound To Danusertib And Inhibiting Monobody Mb2
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2023-09-06 Classification: TRANSFERASE Ligands: EDO, ACT, 627 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: EDO, ACT, 627
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Aura Bound To Danusertib And Activating Monobody Mb1
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2023-09-06 Classification: TRANSFERASE Ligands: EDO, SO4, MES, PO4, PDO, 627 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: EDO, SO4, MES, PO4, PDO, 627
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Structure Of Aurora A (122-403) Bound To Inhibitory Monobody Mb2 And Amppcp
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2019-02-27 Classification: transferase/inhibitor Ligands: ACP |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: ACP
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Pyruvate Decarboxylase From Kluyveromyces Lactis
Organism: Kluyveromyces lactis (strain atcc 8585 / cbs 2359 / dsm 70799 / nbrc 1267 / nrrl y-1140 / wm37)
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2018-08-29 Classification: LYASE Ligands: TPP, MG |
Organism: Kluyveromyces lactis (strain atcc 8585 / cbs 2359 / dsm 70799 / nbrc 1267 / nrrl y-1140 / wm37)
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: TPP, MG
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Pyruvate Decarboxylase From Kluyveromyces Lactis Soaked With Pyruvamide
Organism: Kluyveromyces lactis (strain atcc 8585 / cbs 2359 / dsm 70799 / nbrc 1267 / nrrl y-1140 / wm37)
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2018-08-29 Classification: LYASE Ligands: PY0, TPP, MG, 1PE |
Organism: Kluyveromyces lactis (strain atcc 8585 / cbs 2359 / dsm 70799 / nbrc 1267 / nrrl y-1140 / wm37)
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: PY0, TPP, MG, 1PE
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Structure Of Apo, Dephosphorylated Aurora A (122-403) In An Active Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-06-27 Classification: TRANSFERASE Ligands: P4G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: P4G
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Structure Of Dephosphorylated Aurora A (122-403) Bound To Amppcp In An Active Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-06-27 Classification: TRANSFERASE Ligands: ACP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: ACP, MG
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Structure Of Dephosphorylated Aurora A (122-403) In Complex With Inhibiting Monobody And At9283 In An Inactive Conformation
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2018-06-27 Classification: transferase/inhibitor Ligands: 35R |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: 35R
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Structure Aurora A (122-403) Bound To Activating Monobody Mb1 And Amppcp
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2018-03-14 Classification: TRANSFERASE Ligands: ACP, MG, SO4 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: ACP, MG, SO4
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Crystal Structure Of Adenylate Kinase Ancestor 1 With Zn And Adp Bound
Organism: Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2016-12-28 Classification: TRANSFERASE Ligands: ZN, ADP |
Organism: Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: ZN, ADP
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Crystal Structure Of Adenylate Kinase Ancestor 3 With Zn, Mg And Ap5A Bound
Organism: Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-12-28 Classification: TRANSFERASE Ligands: ZN, AP5, MG |
Organism: Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: ZN, AP5, MG
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Crystal Structure Of Adenylate Kinase Ancestor 4 With Zn And Amp-Adp Bound
Organism: Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2016-12-28 Classification: TRANSFERASE Ligands: ZN, ADP, AMP |
Organism: Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: ZN, ADP, AMP
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Crystal Structure Of Adenylate Kinase Ancestor 4 With Zn, Mg And Ap5A Bound
Organism: Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2016-12-28 Classification: TRANSFERASE Ligands: ZN, AP5, MG |
Organism: Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: ZN, AP5, MG
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Tyrosine Kinase As - A Common Ancestor Of Src And Abl Bound To Gleevec
Organism: Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2015-03-04 Classification: TRANSFERASE Ligands: STI |
Organism: Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2015-03-04
Ligands: STI
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Tyrosine Kinase As - A Common Ancestor Of Src And Abl
Organism: Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2015-02-18 Classification: TRANSFERASE Ligands: ACP |
Organism: Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2015-02-18
Ligands: ACP
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Crystal Structure Of Adenylate Kinase From Aquifex Aeolicus With Mgadp Bound
Organism: Aquifex aeolicus
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2014-12-03 Classification: TRANSFERASE Ligands: ADP, AMP, MG |
Organism: Aquifex aeolicus
Method: X-RAY DIFFRACTION
Release Date: 2014-12-03
Ligands: ADP, AMP, MG
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Cobalt Between Two Adp'S In The Active Site Of Adenylate Kinase
Organism: Aquifex aeolicus
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2014-06-25 Classification: TRANSFERASE Ligands: ADP, CO |
Organism: Aquifex aeolicus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-25
Ligands: ADP, CO
