Search Count: 50
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Structure Of Human Neutrophil Elastase In Complex With A 5,8-Dihydro[1,2,4]Triazolo[4,3-A]Pyrimidin-3(2H)-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.14 Å Release Date: 2025-12-10 Classification: HYDROLASE Ligands: NAG, FUC, A1JN2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-10
Ligands: NAG, FUC, A1JN2
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Degrader-Induced Complex Between Ptpn2 And Crbn-Ddb1
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-09-11 Classification: HYDROLASE Ligands: WO8, ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-09-11
Ligands: WO8, ZN
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Crystal Structure Of Ptpn2 With A Protac
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2024-09-04 Classification: HYDROLASE Ligands: UB0, ACT, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: UB0, ACT, NA
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Structure Of Csf1R Kinase Domain In Complex With Cpd 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2024-05-29 Classification: TRANSFERASE Ligands: A1AE3, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: A1AE3, GOL, SO4
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Structure Of Egfr_D770_N771Insnpg/V948R In Complex With Covalent Inhibitor Osimertinib.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-09-22 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: Q6K, EDO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: Q6K, EDO, CIT
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Crystal Structure Of The First Bromodomain Of Human Brd4 With Benzodiazepine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-09-01 Classification: GENE REGULATION/INHIBITOR Ligands: UDV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-01
Ligands: UDV
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Csf1R Signaling Is A Regulator Of Pathogenesis In Progressive Ms
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: UF4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: UF4
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Crystal Structure Of Fgfr4 Kinase Domain In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-03-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QS7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-25
Ligands: QS7, SO4
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Db-1-264-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2017-08-09 Classification: TRANSCRIPTION/INHIBITOR Ligands: 6TB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: 6TB, EDO
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2015-08-19 Classification: HYDROLASE Ligands: NAG, JJD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-19
Ligands: NAG, JJD
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2015-08-19 Classification: HYDROLASE Ligands: JJS, NAG, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-19
Ligands: JJS, NAG, EPE
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2015-08-19 Classification: HYDROLASE Ligands: NAG, JJX, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-19
Ligands: NAG, JJX, DMS
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-08-19 Classification: HYDROLASE Ligands: JJV, MES, XPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-19
Ligands: JJV, MES, XPE
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Exploitation Of Hydrogen Bonding Constraints And Flat Hydrophobic Energy Landscapes In Pim-1 Kinase Needle Screening And Inhibitor Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2012-03-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0F5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0F5
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Exploitation Of Hydrogen Bonding Constraints And Flat Hydrophobic Energy Landscapes In Pim-1 Kinase Needle Screening And Inhibitor Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2012-03-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0F9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0F9
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Exploitation Of Hydrogen Bonding Constraints And Flat Hydrophobic Energy Landscapes In Pim-1 Kinase Needle Screening And Inhibitor Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2012-03-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0FK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0FK
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Exploitation Of Hydrogen Bonding Constraints And Flat Hydrophobic Energy Landscapes In Pim-1 Kinase Needle Screening And Inhibitor Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2012-03-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0FN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0FN
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Exploitation Of Hydrogen Bonding Constraints And Flat Hydrophobic Energy Landscapes In Pim-1 Kinase Needle Screening And Inhibitor Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2012-03-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0FO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0FO
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Exploitation Of Hydrogen Bonding Constraints And Flat Hydrophobic Energy Landscapes In Pim-1 Kinase Needle Screening And Inhibitor Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2012-03-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0FR, IMD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0FR, IMD
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Exploitation Of Hydrogen Bonding Constraints And Flat Hydrophobic Energy Landscapes In Pim-1 Kinase Needle Screening And Inhibitor Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2012-03-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: IMD, 0FS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: IMD, 0FS