Search Count: 211
![]() |
Jak2 Pseudokinase Domain In Complex With Diaminotriazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2025-11-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1BW6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-05
Ligands: A1BW6
![]() |
Jak2 Pseudokinase Domain In Complex With Diaminotriazole Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-11-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1BXA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-05
Ligands: A1BXA
![]() |
Crystal Structure Of Craf/Mek1 Complex With Plx4720 And Ch5126766
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2025-10-15 Classification: TRANSFERASE Ligands: 324, CHU, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-15
Ligands: 324, CHU, ANP
![]() |
Crystal Structure Of Craf/Mek1 Complex With Plx4720, Ch5126766, And Amppnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2025-10-15 Classification: TRANSFERASE Ligands: 324, CHU, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-15
Ligands: 324, CHU, ANP
![]() |
Cryo-Em Structure Of Craf/Mek1/14-3-3 Complex (Autoinhibited Conformation)
Organism: Homo sapiens, Spodoptera exigua
Method: ELECTRON MICROSCOPY Resolution:3.40 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: AGS, ZN, LCJ |
Organism: Homo sapiens, Spodoptera exigua
Method: ELECTRON MICROSCOPY
Release Date: 2025-09-10
Ligands: AGS, ZN, LCJ
![]() |
Cryo-Em Structure Of Craf/Mek1 Complex (Kinase Domain)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: AGS, MG, LCJ |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-09-10
Ligands: AGS, MG, LCJ
![]() |
Cryo-Em Structure Of Craf/Mek1/14-3-3 Complex (Open Monomer Conformation, Craf Y340D/Y341D Mutant)
Organism: Homo sapiens, Spodoptera exigua
Method: ELECTRON MICROSCOPY Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: AGS, MG, LCJ |
Organism: Homo sapiens, Spodoptera exigua
Method: ELECTRON MICROSCOPY
Release Date: 2025-09-10
Ligands: AGS, MG, LCJ
![]() |
Cryo-Em Structure Of Craf/Mek1 Complex (Kinase Domain, Craf Y340D/Y341D Mutant)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: AGS, MG, LCJ |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-09-10
Ligands: AGS, MG, LCJ
![]() |
Egfr(T790M/V948R) In Complex With Ln2827
Organism: Spodoptera frugiperda
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2025-08-13 Classification: TRANSFERASE Ligands: A1BWA |
Organism: Spodoptera frugiperda
Method: X-RAY DIFFRACTION
Release Date: 2025-08-13
Ligands: A1BWA
![]() |
Egfr(T790M/V948R) In Complex With Ln5461
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2024-08-28 Classification: TRANSFERASE Ligands: MG, ANP, IXC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-08-28
Ligands: MG, ANP, IXC
![]() |
Egfr(T790M/V948R) In Complex With The Allosteric Inhibitor Frf-06-057
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2024-08-28 Classification: TRANSFERASE Ligands: MG, ANP, IXR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-08-28
Ligands: MG, ANP, IXR
![]() |
Egfr(T790M/V948R) Kinase In Complex With Osimertinib And Benzimidazole Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: Q6K, YW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: Q6K, YW5
![]() |
Egfr(T790M/V948R) Kinase In Complex With Benzimidazole Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2024-03-13 Classification: TRANSFERASE Ligands: MG, ANP, YW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-13
Ligands: MG, ANP, YW5
![]() |
Egfr Kinase In Complex With Pyrazolopyrimidine Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-02-14 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: HZ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: HZ6
![]() |
Egfr(T790M/V948R) In Complex With Compound 1 (Ln4503)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-01-17 Classification: TRANSFERASE Ligands: MG, ANP, YA6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: MG, ANP, YA6
![]() |
Egfr(T790M/V948R) In Complex With Compound 2 (Ln5993)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2024-01-17 Classification: TRANSFERASE Ligands: YAA, MG, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: YAA, MG, ANP
![]() |
Egfr Kinase In Complex With Tas6417 (Cln-081)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X9H, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: X9H, CIT
![]() |
Egfr(T790M/V948R) Kinase In Complex With Poziotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R2E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: R2E
![]() |
Egfr Kinase In Complex With Mobocertinib (Tak-788)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R28 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: R28
![]() |
Egfr Kinase In Complex With Poziotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2023-11-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R2E, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-08
Ligands: R2E, CIT
