Search Count: 21
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-02-25 Classification: HYDROLASE Ligands: GDP, A1CRR, MG, CIT |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2026-02-25 Classification: HYDROLASE Ligands: GDP, MG, A1CRV, CIT |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2026-02-25 Classification: HYDROLASE Ligands: GDP, A1CRW, MG, CIT |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-02-25 Classification: HYDROLASE Ligands: GDP, MG, A1CR1, CIT |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2026-02-25 Classification: HYDROLASE Ligands: GDP, MG, A1CR2, CIT |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2026-02-25 Classification: HYDROLASE Ligands: GDP, MG, A1CSD, CIT |
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Crystal Structure Of Atad2A Bromodomain Complexed With H4(1-20)K5Ac Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-12-24 Classification: GENE REGULATION |
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Crystal Structure Of Atad2A Bromodomain Complexed With H3(1-21)K14Ac Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4, CL |
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Crystal Structure Of Atad2A Bromodomain Double Mutant N1063A-Y1064A In Apo Form
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4, CL, GOL |
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Crystal Structure Of Atad2A Bromodomain Complexed With Methyl 3-Amino-5-(3,5-Dimethyl-1,2-Oxazol-4-Yl)Benzoate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4, CL, GOL, 36Z |
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Crystal Structure Of Atad2A Bromodomain Complexed With 3-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-5-[(Phenylsulfonyl)Amino]Benzoicacid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4, GOL, 37N, CL, DMS |
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Crystal Structure Of Apo Atad2A Bromodomain With N1064 Alternate Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2014-12-24 Classification: GENE REGULATION Ligands: SO4 |
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8-Tetrahydropyran-2-Yl Chromans: Highly Selective Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-03 Classification: hydrolase/hydrolase inhibitor Ligands: NI, 3J9 |
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8-Tetrahydropyran-2-Yl Chromans: Highly Selective Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-03 Classification: hydrolase/hydrolase inhibitor Ligands: NI, 3UW |
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8-Tetrahydropyran-2-Yl Chromans: Highly Selective Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-03 Classification: hydrolase/hydrolase inhibitor Ligands: NI, 3UX |
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8-Tetrahydropyran-2-Yl Chromans: Highly Selective Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-12-03 Classification: hydrolase/hydrolase inhibitor Ligands: NI, 3UY |
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Discovery Of 7-Thp Chromans: Bace1 Inhibitors That Reduce A-Beta In The Cns
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-05-14 Classification: hydrolase/hydrolase inhibitor Ligands: NI, 2EX |
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Spirocyclic Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-04-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, 1M4 |
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Spirocyclic Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-04-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, 1M5 |
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Spirocyclic Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (Bace1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-04-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NI, 1M6 |




















