Structural Entry Filters:

Search Count: 10

9YKR image
Crystal Structure Of The Glp (Ehmt1) Set Domain In Complex With Sam And Tng917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.38 Å Release Date: 2026-05-13
Classification: TRANSFERASE
Ligands: ZN, SAM, A1CXM, PEG, SO4, EDO

9YKS image
Crystal Structure Of The G9A (Ehmt2) Set Domain In Complex With Sam And Tng917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.79 Å Release Date: 2026-05-13
Classification: TRANSFERASE
Ligands: ZN, SAM, A1CXM, EDO, GOL

7KKE image
Phosphoinositide 3-Kinase Gamma Bound To A Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.81 Å Release Date: 2021-03-24
Classification: TRANSFERASE/Inhibitor
Ligands: WJV

6C1S image
Phosphoinositide 3-Kinase Gamma Bound To An Pyrrolopyridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.31 Å Release Date: 2018-06-27
Classification: Transferase/Transferase Inhibitor
Ligands: EFV, SO4

5UZJ image
Crystal Structure Of Rock1 Bound To An Aminopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.30 Å Release Date: 2018-03-07
Classification: Transferase/Transferase Inhibitor
Ligands: 8UV

5UZK image
Crystal Structure Of Pka Bound To An Pyrrolo Pyridine Inhibitor
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2018-03-07
Classification: Transferase/Transferase Inhibitor
Ligands: 504

5KKS image
Rock 1 Bound To Azaindole Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.30 Å Release Date: 2017-06-28
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 6U1

5KKT image
Rock 1 Bound To Azaindole Thiazole Piperazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2017-06-28
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 6U2

3B92 image
Novel Thio-Based Tace Inhibitors Part 2: Rational Design, Synthesis And Sar Of Thiol-Contaning Aryl Sufones
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2007-12-18
Classification: HYDROLASE
Ligands: ZN, 440

2OI0 image
Crystal Structure Analysis 0F The Tnf-A Coverting Enzyme (Tace) In Complexed With Aryl-Sulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2007-11-27
Classification: HYDROLASE
Ligands: ZN, 283
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