Search Count: 14
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Crystal Structure Of The Glp (Ehmt1) Set Domain In Complex With Sam And Tng917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2026-05-13 Classification: TRANSFERASE Ligands: ZN, SAM, A1CXM, PEG, SO4, EDO |
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Crystal Structure Of The G9A (Ehmt2) Set Domain In Complex With Sam And Tng917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2026-05-13 Classification: TRANSFERASE Ligands: ZN, SAM, A1CXM, EDO, GOL |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2021-03-24 Classification: TRANSFERASE/Inhibitor Ligands: WJV |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2018-06-27 Classification: Transferase/Transferase Inhibitor Ligands: EFV, SO4 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2018-03-07 Classification: Transferase/Transferase Inhibitor Ligands: 8UV |
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Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-03-07 Classification: Transferase/Transferase Inhibitor Ligands: 504 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6U1 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6U2 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 456 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2015-08-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 43R |
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P5 |
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P6 |
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Novel Thio-Based Tace Inhibitors Part 2: Rational Design, Synthesis And Sar Of Thiol-Contaning Aryl Sufones
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-12-18 Classification: HYDROLASE Ligands: ZN, 440 |
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Crystal Structure Analysis 0F The Tnf-A Coverting Enzyme (Tace) In Complexed With Aryl-Sulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-11-27 Classification: HYDROLASE Ligands: ZN, 283 |














