Search Count: 21
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Brg1 Bromodomain In Complex With Vbc Via Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.17 Å Release Date: 2024-01-17 Classification: GENE REGULATION Ligands: PO4, GOL, VLH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: PO4, GOL, VLH, CL
 |
Vhl/Elongin B/Elongin C Complex With Compound 155
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2024-01-17 Classification: LIGASE Ligands: VL6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: VL6
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Brm (Smarca2) Bromodomain In Complex With Ligand 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2024-01-17 Classification: GENE REGULATION Ligands: ZN, VLC, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-17
Ligands: ZN, VLC, CL
 |
Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: SO4, YR2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: SO4, YR2
 |
Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: SO4, YT2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: SO4, YT2
 |
Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: ZH5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: ZH5
 |
Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2023-10-11 Classification: HYDROLASE/INHIBITOR Ligands: ZJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: ZJX
 |
Crystal Structure Of Tigecycline Degrading Monooxygenase Tet(X4)
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2021-11-10 Classification: OXIDOREDUCTASE Ligands: FDA, GOL |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: FDA, GOL
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Crystal Structure Of Monooxygenase Tet(X4) With Tigecycline
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2021-11-10 Classification: OXIDOREDUCTASE Ligands: FDA, T1C |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2021-11-10
Ligands: FDA, T1C
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Crystal Structure Of The Dna-Binding Domain Of The Nucleoid Occlusion Factor (Noc) Complexed To The Noc-Binding Site (Nbs)
Organism: Bacillus subtilis (strain 168), Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2020-08-05 Classification: DNA BINDING PROTEIN |
Organism: Bacillus subtilis (strain 168), Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2020-08-05
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Crystal Structure Of The Dna Binding Domain Of The Chromosome-Partitioning Protein Parb Complexed To The Centromeric Pars Site
Organism: Caulobacter vibrioides na1000, Caulobacter vibrioides
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-07-15 Classification: DNA BINDING PROTEIN Ligands: GOL |
Organism: Caulobacter vibrioides na1000, Caulobacter vibrioides
Method: X-RAY DIFFRACTION
Release Date: 2020-07-15
Ligands: GOL
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Crystal Structure Of Metallo-Beta-Lactamase Vmb-1
Organism: Vibrio alginolyticus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-11-27 Classification: HYDROLASE Ligands: ZN, CIT |
Organism: Vibrio alginolyticus
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: ZN, CIT
 |
Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9U7
 |
Crebbp Bromodomain In Complex With Cpd8 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2018-03-07 Classification: TRANSFERASE/INHIBITOR Ligands: 9UA, DMS, GOL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UA, DMS, GOL
 |
Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9UD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UD
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Crebbp Bromodomain In Complex With Cpd17 (N,2,7-Trimethyl-2,3-Dihydro-4H-Benzo[B][1,4]Oxazine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: SO4, 9UG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: SO4, 9UG
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Crystal Structure Of Mcr-1, A Phosphoethanolamine Transferase, Extracellular Domain
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2016-12-21 Classification: TRANSFERASE Ligands: ZN |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: ZN
 |
Crystal Structure Of The Bromodomain Of Human Crebbp Bound To Pyrazolopiperidine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XB, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XB, DMS
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Crebbp Bromodomain In Complex With Cpd 44 (3-((5-Acetyl-1-(Cyclopropylmethyl)-4,5,6,7-Tetrahydro-1H-Pyrazolo[4,3-C]Pyridin-3-Yl)Amino)-N-Isopropylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.09 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XG, EDO
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Crebbp Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XH, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XH, EDO, DMS