Search Count: 20
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Probing 3-Amino-2H-Azaindazoles As Allosteric Inhibitors Of The Protein Tyrosine Phosphatase Shp2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2026-06-24 Classification: PEPTIDE BINDING PROTEIN Ligands: A1JWM, ACT, EDO, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-24
Ligands: A1JWM, ACT, EDO, NA
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Mapping The Shp2 Allosteric Pocket With Target-Biased Covalent Fragments
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2026-05-06 Classification: CYTOSOLIC PROTEIN Ligands: EDO, A1JWN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-06
Ligands: EDO, A1JWN
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The Ferm Domain Of Human Moesin With A Bound Peptide Identified By Phage Display
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-03-01 Classification: PROTEIN BINDING Ligands: BR, EDO, B3P |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: BR, EDO, B3P
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The Ferm Domain Of Human Moesin With Two Bound Peptides Identified By Phage Display
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2023-03-01 Classification: PROTEIN BINDING Ligands: ACT, SO4, EDO |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: ACT, SO4, EDO
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The Ferm Domain Of Human Moesin Mutant L281R
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2023-03-01 Classification: PROTEIN BINDING |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
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The Ferm Domain Of Human Moesin Mutant H288A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2023-03-01 Classification: PROTEIN BINDING |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
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Structure Of A T4Ss Effector From Brucella Sp.
Organism: Brucella abortus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2023-01-25 Classification: TOXIN |
Organism: Brucella abortus
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
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Crystal Structure Of Fgfr2 Kinase Domain Gatekeeper Mutant V564F In Complex With Covalent Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2021-02-10 Classification: SIGNALING PROTEIN Ligands: WFD, FLC, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: WFD, FLC, NA
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Crystal Structure Of Fgfr2 Kinase Domain Gatekeeper Mutant V564F In Complex With Covalent Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2021-02-10 Classification: SIGNALING PROTEIN Ligands: WF7, FLC, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: WF7, FLC, GOL
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Cps1 Bound To Allosteric Inhibitor H3B-374
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2021-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 374, ZN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-13
Ligands: 374, ZN, EDO
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Cps1 Bound To Allosteric Inhibitor H3B-193
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-03-18 Classification: LIGASE/LIGASE INHIBITOR Ligands: ZN, Q5A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-18
Ligands: ZN, Q5A
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The High Resolution Structure Of The Ferm Domain And Helical Linker Of Human Moesin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2020-01-29 Classification: PROTEIN BINDING Ligands: ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-29
Ligands: ACT
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The Structure Of The Ferm Domain And Helical Linker Of Human Moesin Bound To A Cd44 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2020-01-29 Classification: PROTEIN BINDING |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-29
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Crystal Structure Of Grasp55 Grasp Domain In Complex With Jam-C C-Terminus
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2017-05-24 Classification: STRUCTURAL PROTEIN/PEPTIDE |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
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Crystal Structure Of Grasp55 Grasp Domain In Complex With Jam-B C-Terminus
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2017-05-24 Classification: STRUCTURAL PROTEIN/PEPTIDE |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
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Crystal Structure Of Archaeal Spt4/5 Bound To The Rnap Clamp Domain
Organism: Pyrococcus furiosus
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2011-03-23 Classification: TRANSCRIPTION Ligands: ZN |
Organism: Pyrococcus furiosus
Method: X-RAY DIFFRACTION
Release Date: 2011-03-23
Ligands: ZN
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Crystal Structure Of Tiox From Micromonospora Sp. Ml1
Organism: Micromonospora sp. ml1
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2010-02-16 Classification: PEPTIDE BINDING PROTEIN |
Organism: Micromonospora sp. ml1
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
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Structure Of The E. Coli Ivy Protein
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2004-11-02 Classification: HYDROLASE INHIBITOR |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2004-11-02
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Ivy:A New Family Of Protein
Organism: Pseudomonas aeruginosa, Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2004-01-14 Classification: HYDROLASE/INHIBITOR |
Organism: Pseudomonas aeruginosa, Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2004-01-14
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Structure Of Ivy Complexed With Its Target, Hewl
Organism: Escherichia coli, Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2003-03-11 Classification: HYDROLASE/INHIBITOR |
Organism: Escherichia coli, Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2003-03-11
