Search Count: 15
![]() |
Structure Of Plasmodium Falciparum 20S Proteasome Bound To An Asparagine-Ethylenediamine Based Inhibitor Tdi6245
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY Resolution:2.86 Å Release Date: 2026-07-29 Classification: HYDROLASE Ligands: A1CRS |
Organism: Plasmodium falciparum
Method: ELECTRON MICROSCOPY
Release Date: 2026-07-29
Ligands: A1CRS
![]() |
Macrocyclic Peptides Tdi5575 That Selectively Inhibit The Mycobacterium Tuberculosis Proteasome
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-04-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: U5Y, CIT, DMF |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2021-04-28
Ligands: U5Y, CIT, DMF
![]() |
Structure Of Mtb Lpd Bound To 010705
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2021-01-27 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: FAD, WPM, GOL |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2021-01-27
Ligands: FAD, WPM, GOL
![]() |
Crystal Structure Of D12 Fab-Atp Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2021-01-13 Classification: IMMUNE SYSTEM Ligands: ATP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-13
Ligands: ATP
![]() |
Crystal Structure Of Switch Ab Fab And Hil6R In Complex With Atp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2021-01-13 Classification: IMMUNE SYSTEM Ligands: SO4, ATP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-13
Ligands: SO4, ATP
![]() |
Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor A85
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMF, M6M, CIT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: DMF, M6M, CIT
![]() |
Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor A86
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMF, M6Y, CIT |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: DMF, M6Y, CIT
![]() |
Crystal Structure Of Mycobacterium Tuberculosis Proteasome In Complex With Phenylimidazole-Based Inhibitor B6
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-10-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: M9G |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: M9G
![]() |
Integrin Alphavbeta3 Ectodomain Bound To Antagonist Tdi-4161
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2019-09-25 Classification: CELL ADHESION Ligands: NAG, MN, JUY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: NAG, MN, JUY
![]() |
Mouse Cgas Bound To The Inhibitor Ru332
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2017-10-11 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: ZN, AE7 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-10-11
Ligands: ZN, AE7
![]() |
Mouse Cgas Bound To The Inhibitor Ru521
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2017-10-11 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: ZN, AEV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-10-11
Ligands: ZN, AEV
![]() |
Mouse Cgas Bound To The Inhibitor Ru365
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2017-08-09 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: ZN, A9Y |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: ZN, A9Y
![]() |
Structure Of Tyk2 With Inhibitor 16: 3-Azanyl-5-[(2~{S})-3-Methylbutan-2-Yl]-7-[1-Methyl-5-(2-Oxidanylpropan-2-Yl)Pyrazol-3-Yl]-1~{H}-Pyrazolo[4,3-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2016-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5U3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-13
Ligands: 5U3
![]() |
Structure Of Tyk2 With Inhibitor 4: 3-Azanyl-5-(2-Methylphenyl)-7-(1-Methylpyrazol-3-Yl)-1~{H}-Pyrazolo[4,3-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2016-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5U4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-13
Ligands: 5U4
![]() |
Crystal Structure Of Human Jnk3 Complexed With An Isoquinolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-09-23 Classification: TRANSFERASE Ligands: 446 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-09-23
Ligands: 446
