Search Count: 17
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Crystal Structure Of Human Vaccinia-Related Kinase 2 (Vrk-2) Bound To Pyridin-Benzenesulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: KJD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: KJD, SO4
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N,N-Dipropyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, ACT, G6J, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: CL, ACT, G6J, SO4, GOL
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Crystal Structure Of The Human Vaccinia-Related Kinase 1 (Vrk1) Bound To An N-Propynyl-N-Isopentyl-Dihydropteridin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-04-04 Classification: Transferase/Transferase Inhibitor Ligands: F87, SO4, ACT, GOL, FCS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: F87, SO4, ACT, GOL, FCS
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N-Methyl-N-Propyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-04-04 Classification: Transferase/Transferase Inhibitor Ligands: SO4, ACT, PG4, FBY, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: SO4, ACT, PG4, FBY, GOL, CL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N-Propynyl-N-Ethyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2018-03-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F8Y, SO4, ACT, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: F8Y, SO4, ACT, GOL, CL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N,N-Dipropynyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-03-21 Classification: Transferase/Transferase Inhibitor Ligands: ACT, F7D, SO4, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: ACT, F7D, SO4, PEG
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A Propynyl-Pteridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-03-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, EA7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: CL, EA7, GOL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A Phenyl-Pteridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-12-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, E8D, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: CL, E8D, SO4, GOL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A Bis-Difluorophenol-Aminopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-12-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: E8V, GOL, CL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: E8V, GOL, CL, SO4
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Crystal Structure Of The Human Camkk2B In Complex With Tae-226
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-12-13 Classification: TRANSFERASE Ligands: BI9, EDO, CL, ACT, NH4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: BI9, EDO, CL, ACT, NH4
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Crystal Structure Of The Human Camkk2B In Complex With Crenolanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-12-13 Classification: TRANSFERASE Ligands: 6T2, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: 6T2, EDO
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Crystal Structure Of The Human Camkk2B In Complex With Bi2526
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-12-13 Classification: TRANSFERASE Ligands: R78, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: R78, ACT
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Crystal Structure Of The Human Camkk2B In Complex With Ap26113-Analog (Alk-In-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-12-13 Classification: TRANSFERASE/TRANSFERASE INHBITOR Ligands: E5J, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: E5J, NA
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A (S)-2-Phenylaminopteridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-12-13 Classification: TRANSFERASE/TRANSFERASE INHBITOR Ligands: SO4, E5M, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-13
Ligands: SO4, E5M, EDO
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Crystal Structure Of The Human Vaccinia-Related Kinase 1 Bound To (R)-2-Phenylaminopteridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-12-06 Classification: transferase/transferase inhibitor Ligands: CL, E1D, EDO, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-06
Ligands: CL, E1D, EDO, SO4, GOL
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Crystal Structure Of The Human Camkk2B Bound To Gsk650394
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-11-29 Classification: TRANSFERASE Ligands: DXV, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-29
Ligands: DXV, FMT
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Crystal Structure Of The Human Camkk2B In Complex With Cp673451
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-11-29 Classification: TRANSFERASE Ligands: 34U, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-29
Ligands: 34U, GOL
