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Crystal Structure Of Human Pin1 Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2026-03-25 Classification: ISOMERASE Ligands: A1D9T |
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Crystal Structure Of Human Pin1 Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2026-03-25 Classification: ISOMERASE Ligands: A1ECA |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2026-03-11 Classification: ISOMERASE Ligands: A1EBR, 1PG |
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Crystal Structure Of Human Pin1 Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2026-03-11 Classification: ISOMERASE Ligands: A1EBS, CIT |
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Human Pin1 (Peptidyl-Prolyl Cis-Trans Isomerase) Catalytic Domain Complexed With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2026-01-21 Classification: ISOMERASE Ligands: A1D9T |
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Human Pin1 (Peptidyl-Prolyl Cis-Trans Isomerase) Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2026-01-21 Classification: ISOMERASE Ligands: A1D9U |
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Crystal Structure Of Human Pin1 Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2026-01-21 Classification: ISOMERASE Ligands: A1D9W, CIT |
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Adp-Ribosyltransferase 1 (Parp1) Catalytic Domain Bound To A Pyrimidine 2,4-Diketone Derivative Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2025-07-09 Classification: TRANSFERASE Ligands: A1D9M, SO4 |
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Mutated Adp-Ribosyltransferase 2 (Parp2) Catalytic Domain Bound To A Pyrimidine 2,4-Diketone Derivative Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-07-09 Classification: TRANSFERASE Ligands: GOL, A1D9M |
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Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-01-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 7TX |
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Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-01-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4YR |
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Structure Of Human Parp1 Catalytic Domain Bound To A Phthalazinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-01-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 7U3 |
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Structure Of Human Parp1 Catalytic Domain Bound To A Benzoimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-01-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 7U6 |
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Structure Of Human Parp1 Catalytic Domain Bound To A Benzoimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-01-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 7U9 |
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Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-01-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 7UL |
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Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-12-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6WX |
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Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2016-12-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6WY |
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Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2016-12-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6X2 |
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Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2016-11-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6WZ |



















