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Search Count: 19

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9JJS image
Crystal Structure Of Human Pin1 Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.52 Å Release Date: 2026-03-25
Classification: ISOMERASE
Ligands: A1D9T

9JJZ image
Crystal Structure Of Human Pin1 Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.61 Å Release Date: 2026-03-25
Classification: ISOMERASE
Ligands: A1ECA

9JF6 image
Crystal Structure Of Human Pin1 In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.96 Å Release Date: 2026-03-11
Classification: ISOMERASE
Ligands: A1EBR, 1PG

9JFH image
Crystal Structure Of Human Pin1 Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.56 Å Release Date: 2026-03-11
Classification: ISOMERASE
Ligands: A1EBS, CIT

9INN image
Human Pin1 (Peptidyl-Prolyl Cis-Trans Isomerase) Catalytic Domain Complexed With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.08 Å Release Date: 2026-01-21
Classification: ISOMERASE
Ligands: A1D9T

9INO image
Human Pin1 (Peptidyl-Prolyl Cis-Trans Isomerase) Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.13 Å Release Date: 2026-01-21
Classification: ISOMERASE
Ligands: A1D9U

9INQ image
Crystal Structure Of Human Pin1 Catalytic Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.17 Å Release Date: 2026-01-21
Classification: ISOMERASE
Ligands: A1D9W, CIT

9ILN image
Adp-Ribosyltransferase 1 (Parp1) Catalytic Domain Bound To A Pyrimidine 2,4-Diketone Derivative Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.49 Å Release Date: 2025-07-09
Classification: TRANSFERASE
Ligands: A1D9M, SO4

9IM8 image
Mutated Adp-Ribosyltransferase 2 (Parp2) Catalytic Domain Bound To A Pyrimidine 2,4-Diketone Derivative Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2025-07-09
Classification: TRANSFERASE
Ligands: GOL, A1D9M

5WRQ image
Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.65 Å Release Date: 2017-01-25
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 7TX

5WRY image
Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2017-01-25
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 4YR

5WRZ image
Structure Of Human Parp1 Catalytic Domain Bound To A Phthalazinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2017-01-25
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 7U3

5WS0 image
Structure Of Human Parp1 Catalytic Domain Bound To A Benzoimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2017-01-25
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 7U6

5WS1 image
Structure Of Human Parp1 Catalytic Domain Bound To A Benzoimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2017-01-25
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 7U9

5WTC image
Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2017-01-25
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 7UL

5KPN image
Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2016-12-21
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 6WX

5KPO image
Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.65 Å Release Date: 2016-12-21
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 6WY

5KPQ image
Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2016-12-14
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 6X2

5KPP image
Structure Of Human Parp1 Catalytic Domain Bound To A Quinazoline-2,4(1H,3H)-Dione Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.33 Å Release Date: 2016-11-30
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 6WZ
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