Search Count: 30
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Crystal Structure Of Human Kras G12D In Complex With Gdp And Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1CZE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1CZE
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Crystal Structure Of Human Kras G12D In Complex With Gdp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1AG3, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1AG3, EDO, SO4
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Crystal Structure Of Human Kras G12D In Complex With Gmppcp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GCP, A1AG3, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GCP, A1AG3, EDO, SO4
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Crystal Structure Of Human Kras G12V In Complex With Gdp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1AG3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1AG3, EDO
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Crystal Structure Of Human Kras G12V In Complex With Gmppcp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GCP, A1AG3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GCP, A1AG3, EDO
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Co-Crystal Structure Of Compound 11 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2023-07-26 Classification: GENE REGULATION Ligands: GOL, FWZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: GOL, FWZ
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Co-Crystal Structure Of Compound 1 In Complex With The Bromodomain Of Human Smarca4 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.73 Å Release Date: 2023-07-26 Classification: GENE REGULATION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
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Crystal Structure Of Rorgt With 3-Cyano-N-(3-{[(3S)-4-(Cyclopentanecarbonyl)-3-Methylpiperazin-1-Yl]Methyl}-5-Fluoro-2-Methylphenyl)Benzamide (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-03-04 Classification: PROTEIN BINDING Ligands: LKY, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: LKY, EDO
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Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
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Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O67 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O67
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5V
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, O5Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: MG, GDP, O5Y
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Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5S
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Imidazopyridazine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-11-09 Classification: transferase/transferase inhibitor Ligands: 6YN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 6YN
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolopyrrolone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-22 Classification: transferase/transferase inhibitor Ligands: 6CD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6CD, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Macrocyclic Quinoxaline-Pyrrolodihydropiperidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-04 Classification: transferase/transferase inhibitor Ligands: 5QO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5QO, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiazolamine-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U5, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiadiazolamine-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U6, GOL