Search Count: 23
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Pcsk9 In Complex With Cyclic Peptide 21
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2026-06-03 Classification: HYDROLASE Ligands: GOL, A1C8P, GOA |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2026-06-03
Ligands: GOL, A1C8P, GOA
 |
Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Indazole Inhibitor Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2024-09-18 Classification: TRANSFERASE Ligands: A1AV4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-18
Ligands: A1AV4, EDO
 |
Structure Of Lrrk2-Chk1 10-Pt. Mutant Complex With Heteroaryl-1H-Indazole Lrrk2 Inhibitor 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2023-02-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: UUF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: UUF
 |
Structure Of Lrrk2-Chk1 10-Pt. Mutant Complex With Heteroaryl-1H-Indazole Lrrk2 Inhibitor 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2023-02-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: UU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: UU6
 |
Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 06
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BVI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: BVI, EDO
 |
Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 09
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BWI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: BWI, EDO
 |
Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BXI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: BXI
 |
Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: L80 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: L80
 |
Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BYL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: BYL
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Pcsk9 In Complex With Compound 19
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2021-11-03 Classification: PROTEIN BINDING,HYDROLASE Ligands: GOL, 89N |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: GOL, 89N
 |
Pcsk9(Deltacrd) In Complex With Cyclic Peptide 35
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2021-11-03 Classification: PROTEIN BINDING,HYDROLASE Ligands: 89N |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: 89N
 |
Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2021-06-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-16
Ligands: YXD
 |
Core Catalytic Domain Of Hiv Integrase In Complex With Virtual Screening Hit
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2020-05-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R2D |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-05-13
Ligands: R2D
 |
Factor Xia In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-05-06 Classification: BLOOD CLOTTING Ligands: CIT, R2Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: CIT, R2Y
 |
Factor Xia In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2020-05-06 Classification: BLOOD CLOTTING Ligands: FLC, R3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: FLC, R3A
 |
Discovery Of Novel Aminobenzisoxazole Derivatives As Orally Available Factor Ixa Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2017-04-26 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: UNL, NA, NHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: UNL, NA, NHE
 |
Discovery Of Novel Aminobenzisoxazole Derivatives As Orally Available Factor Ixa Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-04-26 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 7GQ, NA, NHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: 7GQ, NA, NHE
 |
Development Of A Novel Tricyclic Class Of Potent And Selective Fixa Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2015-11-18 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-18
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Development Of A Novel Class Of Potent And Selective Fixa Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-06-03 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 4M1, NA, NHE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4M1, NA, NHE
 |
Rapid Development Of Two Factor Ixa Inhibitors From Hit To Lead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2015-05-20 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 4K6, NA, NHE, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-20
Ligands: 4K6, NA, NHE, CL