Search Count: 12
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Crystal Structure Of Human Hdac2 In Complex With Tng260
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2025-09-17 Classification: HYDROLASE Ligands: A1B1V, ZN, CA, NHE, EDO, PEG, PGE, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-17
Ligands: A1B1V, ZN, CA, NHE, EDO, PEG, PGE, PG4
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Crystal Structure Of Active Kras-G12C (Gmppnp-Bound) In Complex With Bbo-8520
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-12-18 Classification: ONCOPROTEIN/INHIBITOR Ligands: GNP, MG, Y8N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: GNP, MG, Y8N
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Crystal Structure Of Kras-G12C (Gdp-Bound) In Complex With Bbo-8520
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2024-12-18 Classification: ONCOPROTEIN/INHIBITOR Ligands: GDP, MG, Y8N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: GDP, MG, Y8N
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Structure Of Egfr_D770_N771Insnpg/V948R In Complex With Covalent Inhibitor Osimertinib.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-09-22 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: Q6K, EDO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: Q6K, EDO, CIT
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Egfr With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-06-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, ANP, JBJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-05
Ligands: MG, ANP, JBJ
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Crystal Structure Of Rip1 Kinase In Complex With Gsk547
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.49 Å Release Date: 2018-12-12 Classification: TRANSFERASE Ligands: G4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-12
Ligands: G4W
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Kras G12C In Bound To Quinazoline Based Switch Ii Pocket (Swiip) Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2017-08-23 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: GDP, MG, 91D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-23
Ligands: GDP, MG, 91D
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Kras G12C Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2017-08-23 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: GDP, MG, 91G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-23
Ligands: GDP, MG, 91G
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Egfr Kinase Domain In Complex With Mutant Selective Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2016-06-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, ANP, 57N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: MG, ANP, 57N
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Crystal Structure Of The Jak3 Kinase Domain Covalently Bound To N-(3-(((5-Chloro-2-((2-Methoxy-4-(4-Methylpiperazin-1-Yl)Phenyl)Amino)Pyrimidin-4-Yl)Amino)Methyl)Phenyl)Acrylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2016-02-10 Classification: Transferase/Transferase Inhibitor Ligands: 4LH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 4LH
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Crystal Structure Of Egfr 696-1022 T790M Mutant Covalently Binding To Wz4002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-01-12 Classification: TRANSFERASE Ligands: 0UN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: 0UN
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Escherichia Coli Pyruvate Formate Lyase Large Domain
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2000-05-24 Classification: LYASE/TRANSFERASE |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2000-05-24
