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Cryo-Em Structure Of Ternary Complex Bcl6-Crbn-Ddb1 With Bms-986458 (Local Refined), A Potent And Selective Bcl6 Ligand Directed Degrader (Ldd)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.09 Å Release Date: 2026-02-18 Classification: LIGASE Ligands: A1CTU, ZN |
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Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, CL, A1BLT, CIT |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, NI, A1BLT |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, A1BLO |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, SO4, A1BLN |
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Bruton'S Tyrosine Kinase In Complex With N-[(2R)-1-[(3R)-3-(Methylcarbamoyl)-1H,2H,3H,4H,9H-Pyrido[3,4-B]Indol-2-Yl]-3-(3-Methylphenyl)-1-Oxopropan-2-Yl]-1H-Indazole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-01-31 Classification: TRANSFERASE Ligands: UQX, NA, CL, SO4, EDO |
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Bruton'S Tyrosine Kinase In Complex With N-[(2R)-1-[(3R)-3-(Methylcarbamoyl)-1H,2H,3H,4H,9H-Pyrido[3,4-B]Indol-2-Yl]-3-(3-Methylphenyl)-1-Oxopropan-2-Yl]-1H-Indazole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-01-31 Classification: TRANSFERASE Ligands: UP9, EDO, CL, IOD |







