Search Count: 26
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 4).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.58 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YO4, YNZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YO4, YNZ
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket (Compound 5).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YOR, YNZ, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YOR, YNZ, CL
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Pi3Ka H1047R Co-Crystal Structure With Inhibitors In Two Cryptic Pockets (Compounds 4 And 5).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.35 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YO4, YOR, YNZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YO4, YOR, YNZ
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 12).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: 1LT, YQB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: 1LT, YQB
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Pi3Ka H1047R Co-Crystal Structure With Inhibitor In Cryptic Pocket Near H1047R (Compound 7).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2024-03-20 Classification: SIGNALING PROTEIN Ligands: YQ2, 1LT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-20
Ligands: YQ2, 1LT
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Crystal Structure Of Human Il-17A Cytokine In Complex With Macrocycle
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2023-12-06 Classification: CYTOKINE Ligands: UTF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: UTF
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Complex Of Pd-L1 With Vhh6
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-06-14 Classification: IMMUNE SYSTEM Ligands: PEG, ACY, OXM, EDO, FMT, PG4 |
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: PEG, ACY, OXM, EDO, FMT, PG4
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Complex Of Pd-L1 With Vhh1
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-06-14 Classification: IMMUNE SYSTEM Ligands: MG |
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: MG
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Prmt5/Mep50 Crystal Structure With Mta And An Achiral, Class 1, Non-Atropisomeric Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2022-08-17 Classification: TRANSFERASE Ligands: NXF, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-17
Ligands: NXF, MTA
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Prmt5/Mep50 Crystal Structure With Sinefungin Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2022-03-16 Classification: TRANSFERASE/INHIBITOR Ligands: SFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: SFG
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Prmt5/Mep50 Crystal Structure With Mta And Phthalazinone Fragment Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2022-01-26 Classification: TRANSFERASE Ligands: CL, NA, EDO, 81X, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: CL, NA, EDO, 81X, MTA
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Prmt5/Mep50 Crystal Structure With Mta And A Phthalazinone Inhibitor Bound (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 84W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 84W
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Prmt5/Mep50 Crystal Structure With Mta And A Phthalazinone Inhibitor Bound (Compound (M)-31)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 85E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 85E
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Prmt5/Mep50 Crystal Structure With Mta And Mrtx-1719 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: MTA, 85K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: MTA, 85K
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Prmt5/Mep50 With Compound 30 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: 97L, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: 97L, MTA
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Prmt5/Mep50 With Compound 29 Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-01-26 Classification: TRANSFERASE/INHIBITOR Ligands: 97X, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-26
Ligands: 97X, MTA
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Solution Structure Of The N-Terminal Region Of Dkk4
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2018-06-13 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2018-06-13
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Crystal Structure Of Fcrn At Ph3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-05-30 Classification: IMMUNE SYSTEM Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: GOL
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Crystal Structure Of Fcrn Bound To Ucb-84
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-30 Classification: IMMUNE SYSTEM Ligands: CYS, ER7, GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: CYS, ER7, GOL, PEG
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Crystal Structure Of Fcrn Bound To Ucb-303
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-05-30 Classification: IMMUNE SYSTEM Ligands: EQY, NAG, GOL, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: EQY, NAG, GOL, CIT
