Search Count: 15
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Cryoem Structure Of Prmt5 Bound To Covalent Pbm-Site Inhibitor Brd-6988
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-03-17 Classification: TRANSFERASE/INHIBITOR Ligands: YJG |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2021-03-17
Ligands: YJG
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Prmt5 Complex Bound To Covalent Pbm Inhibitor Brd6711
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2020-11-25 Classification: SPLICING/TRANSFERASE Ligands: QN4, CL, SFG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: QN4, CL, SFG, GOL
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Crystal Structure Of Danio Rerio Histone Deacetylase 6 Catalytic Domain 2 In Complex With Cyclohexenylhydroxamate
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2018-05-30 Classification: HYDROLASE Ligands: ZN, K, CL, FBM, EDO, PEG |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: ZN, K, CL, FBM, EDO, PEG
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Crystal Structure Of Danio Rerio Histone Deacetylase 6 Catalytic Domain 2 In Complex With Cyclohexylhydroxamate
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2018-05-30 Classification: HYDROLASE Ligands: ZN, K, F9P |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: ZN, K, F9P
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Crystal Structure Of Danio Rerio Histone Deacetylase 6 Catalytic Domain 2 In Complex With Phenylhydroxamate
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2018-05-30 Classification: HYDROLASE Ligands: ZN, K, BHO, EDO |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: ZN, K, BHO, EDO
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Crystal Structure Of Danio Rerio Histone Deacetylase 6 Catalytic Domain 2 In Complex With Cyclopentenylhydroxamate
Organism: Danio rerio
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-05-30 Classification: HYDROLASE Ligands: ZN, K, FBJ, EDO |
Organism: Danio rerio
Method: X-RAY DIFFRACTION
Release Date: 2018-05-30
Ligands: ZN, K, FBJ, EDO
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VK
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0705
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VL
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Glycogen Synthase Kinase 3 Beta Complexed With Brd3731
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VM
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Exploiting An Asp-Glu Switch In Glycogen Synthase Kinase 3 To Design Paralog Selective Inhibitors For Use In Acute Myeloid Leukemia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 6VL
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Crystal Structure Of Gsk-3Beta Complexed With Pf-04802367, A Highly Selective Brain-Penetrant Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-09-21 Classification: TRANSFERASE Ligands: 6QH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6QH, SO4
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Hdac2 With Ligand Brd4884
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2016-08-31 Classification: HYDROLASE Ligands: ZN, CA, IWX, PG5, PGE, PEG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: ZN, CA, IWX, PG5, PGE, PEG, PG4
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Hdac2 With Ligand Brd7232
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2016-08-31 Classification: HYDROLASE Ligands: ZN, CA, 6EZ, PEG, PG4, PG5, PGE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: ZN, CA, 6EZ, PEG, PG4, PG5, PGE, EDO
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X-Ray Crystal Structure Of Gsk3B In Complex With Chir99021
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65C, MG, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 65C, MG, MES
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X-Ray Crystal Structure Of Gsk3B In Complex With Brd3937
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 65A
