Search Count: 25
 |
Mettl1 Bound To The Sam Competitive Small Molecule Inhibitor Stm9005
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2026-08-26 Classification: TRANSFERASE Ligands: A1JKJ, SO4, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-26
Ligands: A1JKJ, SO4, EDO, CL
 |
Mettl3-Mettl14 Heterodimer Bound To The Sam Competitive Small Molecule Inhibitor Stm2457
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2021-04-14 Classification: RNA BINDING PROTEIN Ligands: V22, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: V22, DMS
 |
Hbo1 Is Required For The Maintenance Of Leukaemia Stem Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2019-12-25 Classification: antitumor protein/inhibitor Ligands: ZN, GOL, JAV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: ZN, GOL, JAV
 |
Hbo1 Is Required For The Maintenance Of Leukaemia Stem Cells
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2019-12-25 Classification: antitumor protein/transferase Ligands: ZN, ACO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: ZN, ACO
 |
Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9U7
 |
Crebbp Bromodomain In Complex With Cpd8 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2018-03-07 Classification: TRANSFERASE/INHIBITOR Ligands: 9UA, DMS, GOL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UA, DMS, GOL
 |
Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9UD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UD
 |
Crebbp Bromodomain In Complex With Cpd17 (N,2,7-Trimethyl-2,3-Dihydro-4H-Benzo[B][1,4]Oxazine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: SO4, 9UG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: SO4, 9UG
 |
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Bromosporine (Bsp)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-10-19 Classification: TRANSCRIPTION Ligands: EDO, BMF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-19
Ligands: EDO, BMF
 |
Crystal Structure Of The Second Bromodomain Of Human Taf1L In Complex With Bromosporine (Bsp)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-10-19 Classification: TRANSCRIPTION Ligands: BMF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-19
Ligands: BMF
 |
Crystal Structure Of The Bromodomain Of Human Brd9 In Complex With Bromosporine (Bsp)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-10-19 Classification: TRANSCRIPTION Ligands: BMF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-19
Ligands: BMF
 |
Lactate Dehydrogenase A In Complex With A Trisubstituted Piperidine-2,4-Dione Inhibitor Gne-140
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-18 Classification: Oxidoreductase/Oxidoreductase Inhibitor Ligands: NAD, SO4, GN0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: NAD, SO4, GN0
 |
Crystal Structure Of The Cbp Bromodomain In Complex With Cpi098
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 986, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 986, EDO
 |
Crystal Structure Of The Cbp Bromodomain In Complex With Cpi703
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING Ligands: 58N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 58N
 |
Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Sorafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BAX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: BAX
 |
Egfr Kinase Domain Mutant "Tmlr" With A Pyrazolopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 63M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 63M
 |
Egfr Kinase Domain Mutant "Tmlr" With A Imidazopyridinyl-Aminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 63N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: SO4, 63N
 |
Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Az628
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B1E, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: B1E, PEG
 |
Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Dabrafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: P06
 |
Crystal Structure Of Mek1 Kinase Bound To Gdc0973
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-08-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ANP, MG, EUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: ANP, MG, EUI