Search Count: 21
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Crystal Structure Of Cdk9-Cyclin T1 Bound By Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2021-10-27 Classification: TRANSFERASE Ligands: UT5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-27
Ligands: UT5
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn012042
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: XRM, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: XRM, CL, EDO
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn011980
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: YFG, CL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: YFG, CL, GOL
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn012759
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2021-03-24 Classification: TRANSFERASE/Inhibitor Ligands: XBA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: XBA, EDO
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2021-03-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: TZ7, EDO, PEG, GOL, SO4, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: TZ7, EDO, PEG, GOL, SO4, PGE
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2021-03-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: FDR, EDO, TYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: FDR, EDO, TYG, GOL
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Cdk9-Cyclin-T1 Complex Bound By Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.37 Å Release Date: 2020-12-23 Classification: TRANSFERASE Ligands: Q6E, TRS, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: Q6E, TRS, PO4
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Human Poly(Adp-Ribose) Polymerase 12, Catalytic Fragment With Four Point Mutations In Complex With Rbn-2397
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-12-16 Classification: TRANSFERASE Ligands: QO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: QO4, CL
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Human Parp16 In Complex With Rbn010860
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2020-10-07 Classification: TRANSFERASE Ligands: T9D, CIT, GOL, EDO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: T9D, CIT, GOL, EDO, PEG
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Human Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-04-29 Classification: TRANSFERASE Ligands: LKT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: LKT, EDO
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Human Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-04-29 Classification: TRANSFERASE Ligands: LKQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: LKQ
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Chk1 Kinase In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: SO4, D4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: SO4, D4Q
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Chk1 Kinase In Complex With Compound 44
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: D58, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D58, SO4
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Chk1 Kinase In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: D4Z, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D4Z, SO4
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Human Jak1 Kinase In Complex With Compound 30 At 2.30 Angstroms Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-11-25 Classification: TRANSFERASE Ligands: PEG, 5JG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: PEG, 5JG
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Ephb4 Kinase Domain Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2013-02-27 Classification: TRANSFERASE Ligands: 32W, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: 32W, MG
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Braf In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2013-02-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 10Z, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: 10Z, CL
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, YDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, YDI
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, GOL, YDK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, GOL, YDK
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2012-01-25 Classification: TRANSFERASE Ligands: YDJ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-25
Ligands: YDJ, PO4
