Structural Entry Filters:

Search Count: 21

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7NWK image
Crystal Structure Of Cdk9-Cyclin T1 Bound By Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.81 Å Release Date: 2021-10-27
Classification: TRANSFERASE
Ligands: UT5

7L9Y image
Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn012042

7LUN image
Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn011980

6WE2 image
Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn012759

6WE3 image
Human Parp14 (Artd8), Catalytic Fragment In Complex With Compound 3

6WE4 image
Human Parp14 (Artd8), Catalytic Fragment In Complex With Compound 2

6Z45 image
Cdk9-Cyclin-T1 Complex Bound By Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.37 Å Release Date: 2020-12-23
Classification: TRANSFERASE
Ligands: Q6E, TRS, PO4

6V3W image
Human Poly(Adp-Ribose) Polymerase 12, Catalytic Fragment With Four Point Mutations In Complex With Rbn-2397
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.04 Å Release Date: 2020-12-16
Classification: TRANSFERASE
Ligands: QO4, CL

6W65 image
Human Parp16 In Complex With Rbn010860
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.13 Å Release Date: 2020-10-07
Classification: TRANSFERASE
Ligands: T9D, CIT, GOL, EDO, PEG

6SM8 image
Human Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2020-04-29
Classification: TRANSFERASE
Ligands: LKT, EDO

6SMB image
Human Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.04 Å Release Date: 2020-04-29
Classification: TRANSFERASE
Ligands: LKQ

6FC8 image
Chk1 Kinase In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.61 Å Release Date: 2018-01-17
Classification: TRANSFERASE
Ligands: SO4, D4Q

6FCF image
Chk1 Kinase In Complex With Compound 44
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2018-01-17
Classification: TRANSFERASE
Ligands: D58, SO4

6FCK image
Chk1 Kinase In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2018-01-17
Classification: TRANSFERASE
Ligands: D4Z, SO4

5E1E image
Human Jak1 Kinase In Complex With Compound 30 At 2.30 Angstroms Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2015-11-25
Classification: TRANSFERASE
Ligands: PEG, 5JG

4BB4 image
Ephb4 Kinase Domain Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.65 Å Release Date: 2013-02-27
Classification: TRANSFERASE
Ligands: 32W, MG

4H58 image
Braf In Complex With Compound 3

2YDI image
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2012-04-04
Classification: TRANSFERASE
Ligands: SO4, YDI

2YDK image
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2012-04-04
Classification: TRANSFERASE
Ligands: SO4, GOL, YDK

2YDJ image
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2012-01-25
Classification: TRANSFERASE
Ligands: YDJ, PO4
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