Search Count: 90
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Structure Of Gpr61 Bound To Inverse Agonist Compound 15
Organism: Homo sapiens, Lama glama
Method: ELECTRON MICROSCOPY Resolution:3.08 Å Release Date: 2026-03-25 Classification: SIGNALING PROTEIN Ligands: A1CWB |
Organism: Homo sapiens, Lama glama
Method: ELECTRON MICROSCOPY
Release Date: 2026-03-25
Ligands: A1CWB
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Pad2 With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-07-30 Classification: HYDROLASE Ligands: A1CE0, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: A1CE0, CA
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2025-05-28 Classification: HYDROLASE Ligands: CA, A1A8O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1A8O
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Inhibiting Peptidylarginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, A1BZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1BZK
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1A9P, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1A9P, 3YZ
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Crystal Structure Of The Human Pad2 Protein Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: A1AJA, ACT, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1AJA, ACT, CA
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Crystal Structure Of The Human Pad2 Protein Bound To Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: MPD, A1AJB, ACT, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: MPD, A1AJB, ACT, CA
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Crystal Structure Of The Human Pad2 Protein Bound To Small Molecule
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2024-10-09 Classification: HYDROLASE Ligands: ACT, CA, A1AJC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: ACT, CA, A1AJC
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 5 Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: LKY, 4Y5, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: LKY, 4Y5, SO4
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 6A Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: XNR, 4Y5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: XNR, 4Y5
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 8 Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: XO5, XNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: XO5, XNX
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Vanin-1 Complexed With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2022-01-12 Classification: HYDROLASE Ligands: NAG, 9TC, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: NAG, 9TC, NA
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Vanin-1 Complexed With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2022-01-12 Classification: HYDROLASE Ligands: NAG, 9SS, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: NAG, 9SS, NA
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Vanin-1 Complexed With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2022-01-12 Classification: HYDROLASE Ligands: NAG, 9S5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: NAG, 9S5
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Crystal Structure Of Jak2 With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWP
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Crystal Structure Of Tyk2 With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWP
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Crystal Structure Of Tyk2 With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2020-11-25 Classification: TRANSFERASE Ligands: UWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: UWM
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Crystal Structure Of Tyk2 Kinase With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R5D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R5D
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Crystal Structure Of Tyk2 Kinase With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4Y
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Crystal Structure Of Tyk2 Kinase With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2020-04-08 Classification: TRANSFERASE/INHIBITOR Ligands: R4V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R4V
