Search Count: 26
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Crystal Structure Of C-Met-D1228N In Complex With Kin-7615
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: A1AB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: A1AB1
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The X-Ray Co-Crystal Structure Of Human Fgfr3 And Kin-3248
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2024-02-07 Classification: TRANSFERASE/INHIBITOR Ligands: MLT, WGF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: MLT, WGF
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The X-Ray Co-Crystal Structure Of Human Fgfr3 And Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2024-02-07 Classification: TRANSFERASE/INHIBITOR Ligands: CL, WIQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: CL, WIQ
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The X-Ray Co-Crystal Structure Of Human Fgfr3 V555M And Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2024-02-07 Classification: TRANSFERASE/INHIBITOR Ligands: SO4, WIQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: SO4, WIQ, EDO
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Crystal Structure Of Lysine Specific Demethylase 1 (Lsd1) With Cc-90011
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2020-10-21 Classification: FLAVOPROTEIN Ligands: V0Y, FAD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: V0Y, FAD
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Crystal Structure Of Kdm4 With The Small Molecule Inhibitor Qc6352
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-09-27 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, 9DJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NI, ZN, 9DJ
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Crystal Structure Of Human Kdm4 With Small Molecule Inhibitor Qc5714
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-09-27 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, 9FJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NI, ZN, 9FJ
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Crystal Structure Of The Fifth Bromodomain Of Human Pb1 In Complex With 1-Ethylisochromeno[3,4-C]Pyrazol-5(2H)-One) Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: 64C, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 64C, EDO
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Crystal Structure Of The Fifth Bromodomain Of Human Pb1 In Complex With 1-Propylisochromeno[3,4-C]Pyrazol-5(2H)-One) Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: 64E, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 64E, EDO, SO4
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Crystal Structure Of The Fifth Bromodomain Of Human Pb1 In Complex With 1-Butylisochromeno[3,4-C]Pyrazol-5(2H)-One) Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: EDO, 64F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: EDO, 64F
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Crystal Structure Of The Fifth Bromodomain Of Human Polybromo (Pb1) In Complex With 1-Methylisochromeno[3,4-C]Pyrazol-5(3H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2016-06-29 Classification: TRANSCRIPTION Ligands: 6BL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 6BL
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Crystal Structure Of The Fifth Bromodomain Of Human Polybromo (Pb1) In Complex With 2-(3,4-Dihydroxyphenyl)-5,7-Dihydroxy-4H-Chromen-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-29 Classification: TRANSCRIPTION Ligands: K, CIT, LU2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: K, CIT, LU2
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Crystal Structure Of The Fifth Bromodomain Of Human Polybromo (Pb1) In Complex With 2-(3,4-Dihydroxyphenyl)-5-Hydroxy-4H-Chromen-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-06-29 Classification: TRANSCRIPTION Ligands: 6BK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 6BK
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Fragment-Based Discovery Of A Small Molecule Reversible Inhibitor Of Bruton'S Tyrosine Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: IMD, IPA, EDO, 4L6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, EDO, 4L6
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Crystal Structure Of Bruton'S Tyrosine Kinase Bound To A Cinnoline Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2015-07-01 Classification: Transferase/Transferase Inhibitor Ligands: IMD, IPA, DMS, 4RU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, DMS, 4RU
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Crystal Structure Of Bruton'S Tyrosine Kinase In Complex With A Substituted Cinnoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-07-01 Classification: Transferase/Transferase Inhibitor Ligands: IMD, IPA, DMS, 4RV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, DMS, 4RV
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Dimeric Horse Myoglobin
Organism: Equus caballus
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2012-09-12 Classification: OXYGEN STORAGE Ligands: O, HEM |
Organism: Equus caballus
Method: X-RAY DIFFRACTION
Release Date: 2012-09-12
Ligands: O, HEM
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Crystal Structure Of The Human Kinase And Rnase Domains In Complex With Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-02-23 Classification: HYDROLASE, Transferase Ligands: MG, ADP, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-23
Ligands: MG, ADP, SO4
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Crystal Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek 1) In Complex With Ligand And Mgatp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ATP, MG, IZG, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-23
Ligands: ATP, MG, IZG, ACT
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Crystal Structure Of Actin Capping Protein In Complex With Carmil Fragment
Organism: Gallus gallus, Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2010-11-17 Classification: PROTEIN BINDING |
Organism: Gallus gallus, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-11-17
