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8VI1 image
Crystal Structure Of C-Met-D1228N In Complex With Kin-7615
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.11 Å Release Date: 2025-04-02
Classification: TRANSFERASE
Ligands: A1AB1

8UDT image
The X-Ray Co-Crystal Structure Of Human Fgfr3 And Kin-3248
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.83 Å Release Date: 2024-02-07
Classification: TRANSFERASE/INHIBITOR
Ligands: MLT, WGF

8UDU image
The X-Ray Co-Crystal Structure Of Human Fgfr3 And Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.74 Å Release Date: 2024-02-07
Classification: TRANSFERASE/INHIBITOR
Ligands: CL, WIQ

8UDV image
The X-Ray Co-Crystal Structure Of Human Fgfr3 V555M And Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.35 Å Release Date: 2024-02-07
Classification: TRANSFERASE/INHIBITOR
Ligands: SO4, WIQ, EDO

6W4K image
Crystal Structure Of Lysine Specific Demethylase 1 (Lsd1) With Cc-90011
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.93 Å Release Date: 2020-10-21
Classification: FLAVOPROTEIN
Ligands: V0Y, FAD

5VGI image
Crystal Structure Of Kdm4 With The Small Molecule Inhibitor Qc6352
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.07 Å Release Date: 2017-09-27
Classification: OXIDOREDUCTASE/INHIBITOR
Ligands: NI, ZN, 9DJ

5VMP image
Crystal Structure Of Human Kdm4 With Small Molecule Inhibitor Qc5714
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.48 Å Release Date: 2017-09-27
Classification: OXIDOREDUCTASE/INHIBITOR
Ligands: NI, ZN, 9FJ

5HRV image
Crystal Structure Of The Fifth Bromodomain Of Human Pb1 In Complex With 1-Ethylisochromeno[3,4-C]Pyrazol-5(2H)-One) Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2016-10-12
Classification: TRANSCRIPTION
Ligands: 64C, EDO

5HRW image
Crystal Structure Of The Fifth Bromodomain Of Human Pb1 In Complex With 1-Propylisochromeno[3,4-C]Pyrazol-5(2H)-One) Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2016-10-12
Classification: TRANSCRIPTION
Ligands: 64E, EDO, SO4

5HRX image
Crystal Structure Of The Fifth Bromodomain Of Human Pb1 In Complex With 1-Butylisochromeno[3,4-C]Pyrazol-5(2H)-One) Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.73 Å Release Date: 2016-10-12
Classification: TRANSCRIPTION
Ligands: EDO, 64F

5II1 image
Crystal Structure Of The Fifth Bromodomain Of Human Polybromo (Pb1) In Complex With 1-Methylisochromeno[3,4-C]Pyrazol-5(3H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.02 Å Release Date: 2016-06-29
Classification: TRANSCRIPTION
Ligands: 6BL

5II2 image
Crystal Structure Of The Fifth Bromodomain Of Human Polybromo (Pb1) In Complex With 2-(3,4-Dihydroxyphenyl)-5,7-Dihydroxy-4H-Chromen-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2016-06-29
Classification: TRANSCRIPTION
Ligands: K, CIT, LU2

5IID image
Crystal Structure Of The Fifth Bromodomain Of Human Polybromo (Pb1) In Complex With 2-(3,4-Dihydroxyphenyl)-5-Hydroxy-4H-Chromen-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2016-06-29
Classification: TRANSCRIPTION
Ligands: 6BK

4Z3V image
Fragment-Based Discovery Of A Small Molecule Reversible Inhibitor Of Bruton'S Tyrosine Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2015-07-01
Classification: TRANSFERASE
Ligands: IMD, IPA, EDO, 4L6

4ZLY image
Crystal Structure Of Bruton'S Tyrosine Kinase Bound To A Cinnoline Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.65 Å Release Date: 2015-07-01
Classification: Transferase/Transferase Inhibitor
Ligands: IMD, IPA, DMS, 4RU

4ZLZ image
Crystal Structure Of Bruton'S Tyrosine Kinase In Complex With A Substituted Cinnoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2015-07-01
Classification: Transferase/Transferase Inhibitor
Ligands: IMD, IPA, DMS, 4RV

3VM9 image
Dimeric Horse Myoglobin
Organism: Equus caballus
Method: X-RAY DIFFRACTION
Resolution:1.05 Å Release Date: 2012-09-12
Classification: OXYGEN STORAGE
Ligands: O, HEM

3P23 image
Crystal Structure Of The Human Kinase And Rnase Domains In Complex With Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2011-02-23
Classification: HYDROLASE, Transferase
Ligands: MG, ADP, SO4

3PP1 image
Crystal Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek 1) In Complex With Ligand And Mgatp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2011-02-23
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: ATP, MG, IZG, ACT

3AAE image
Crystal Structure Of Actin Capping Protein In Complex With Carmil Fragment
Organism: Gallus gallus, Mus musculus
Method: X-RAY DIFFRACTION
Resolution:3.30 Å Release Date: 2010-11-17
Classification: PROTEIN BINDING
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